HIGH-RESOLUTION X-RAY ANALYSES OF RENIN INHIBITOR-ASPARTIC PROTEINASE COMPLEXES

被引:133
作者
FOUNDLING, SI
COOPER, J
WATSON, FE
CLEASBY, A
PEARL, LH
SIBANDA, BL
HEMMINGS, A
WOOD, SP
BLUNDELL, TL
VALLER, MJ
NOREY, CG
KAY, J
BOGER, J
DUNN, BM
LECKIE, BJ
JONES, DM
ATRASH, B
HALLETT, A
SZELKE, M
机构
[1] UNIV WALES UNIV COLL CARDIFF,DEPT BIOCHEM,CARDIFF CF1 1XL,S GLAM,WALES
[2] MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
[3] UNIV FLORIDA,COLL MED,DEPT BIOCHEM & MOLEC BIOL,GAINESVILLE,FL 32610
[4] WESTERN INFIRM,BLOOD PRESSURE UNIT,GLASGOW G11 6NT,SCOTLAND
[5] ROYAL POSTGRAD MED SCH,LONDON W12 0HS,ENGLAND
关键词
D O I
10.1038/327349a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:349 / 352
页数:4
相关论文
共 28 条
[11]  
HALLETT A, 1985, ASPARTIC PROTEINASES, P467
[12]   RESTRAINED STRUCTURE-FACTOR LEAST-SQUARES REFINEMENT OF PROTEIN STRUCTURES USING A VECTOR PROCESSING COMPUTER [J].
HANEEF, I ;
MOSS, DS ;
STANFORD, MJ ;
BORKAKOTI, N .
ACTA CRYSTALLOGRAPHICA SECTION A, 1985, 41 (SEP) :426-433
[13]   MOLECULAR-STRUCTURE OF AN ASPARTIC PROTEINASE ZYMOGEN, PORCINE PEPSINOGEN, AT 1.8 A RESOLUTION [J].
JAMES, MNG ;
SIELECKI, AR .
NATURE, 1986, 319 (6048) :33-38
[14]   CONFORMATIONAL FLEXIBILITY IN THE ACTIVE-SITES OF ASPARTYL PROTEINASES REVEALED BY A PEPSTATIN FRAGMENT BINDING TO PENICILLOPEPSIN [J].
JAMES, MNG ;
SIELECKI, A ;
SALITURO, F ;
RICH, DH ;
HOFMANN, T .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (20) :6137-6141
[15]   STRUCTURE AND REFINEMENT OF PENICILLOPEPSIN AT 1.8-A RESOLUTION [J].
JAMES, MNG ;
SIELECKI, AR .
JOURNAL OF MOLECULAR BIOLOGY, 1983, 163 (02) :299-361
[16]  
JONES AT, 1978, J APPL CRYSTALLOGR, V11, P268
[17]   PEPTIDE INHIBITORS OF RENIN-ANGIOTENSIN SYSTEM [J].
KOKUBU, T ;
UEDA, E ;
FUJIMOTO, S ;
HIWADA, K ;
KATO, A ;
AKUTSU, H ;
YAMAMURA, Y ;
SAITO, S ;
MIZOGUCH.T .
NATURE, 1968, 217 (5127) :456-&
[18]  
NAVIA MA, 1984, J BIOL CHEM, V259, P2714
[19]   THE ACTIVE-SITE OF ASPARTIC PROTEINASES [J].
PEARL, L ;
BLUNDELL, T .
FEBS LETTERS, 1984, 174 (01) :96-101
[20]  
PEDERSEN VB, IN PRESS BIOCHEMISTR