URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS

被引:624
作者
BRAESTRUP, C
NIELSEN, M
OLSEN, CE
机构
[1] SCT HANS HOSP,DK-4000 ROSKILDE,DENMARK
[2] ROYAL VET & AGR UNIV,DK-1871 COPENHAGEN,DENMARK
来源
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES | 1980年 / 77卷 / 04期
关键词
D O I
10.1073/pnas.77.4.2288
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:2288 / 2292
页数:5
相关论文
共 52 条
[31]  
MAELICKE A, 1977, J BIOL CHEM, V252, P4811
[32]   5-METHYLTETRAHYDROFOLIC ACID AS A MEDIATOR IN FORMATION OF PYRIDOINDOLES [J].
MANDEL, LR ;
ROSEGAY, A ;
WALKER, RW ;
VANDENHEUVEL, WJ ;
ROKACH, J .
SCIENCE, 1974, 186 (4165) :741-743
[33]   CONSTITUENTS OF NAUCLEA-DIDERRICHII .2. ISOLATION AND CLASSIFICATION OF CONSTITUENTS - SIMPLE BETA-CARBOLINE AND PYRIDINE ALKALOIDS [J].
MCLEAN, S ;
MURRAY, DG .
CANADIAN JOURNAL OF CHEMISTRY, 1972, 50 (10) :1478-&
[34]   BENZODIAZEPINE RECEPTOR IN NORMAL AND PATHOLOGICAL HUMAN-BRAIN [J].
MOHLER, H ;
OKADA, T .
BRITISH JOURNAL OF PSYCHIATRY, 1978, 133 (SEP) :261-268
[35]   NICOTINAMIDE IS A BRAIN CONSTITUENT WITH BENZODIAZEPINE-LIKE ACTIONS [J].
MOHLER, H ;
POLC, P ;
CUMIN, R ;
PIERI, L ;
KETTLER, R .
NATURE, 1979, 278 (5704) :563-565
[36]   PROPERTIES OF DIAZEPAM-H-3 BINDING TO BENZODIAZEPINE RECEPTORS IN RAT CEREBRAL-CORTEX [J].
MOHLER, H ;
OKADA, T .
LIFE SCIENCES, 1977, 20 (12) :2101-2110
[37]   BENZODIAZEPINE RECEPTOR - DEMONSTRATION IN CENTRAL NERVOUS-SYSTEM [J].
MOHLER, H ;
OKADA, T .
SCIENCE, 1977, 198 (4319) :849-851
[38]   EVIDENCE FOR A LATE EVOLUTIONARY APPEARANCE OF BRAIN-SPECIFIC BENZODIAZEPINE RECEPTORS - INVESTIGATION OF 18 VERTEBRATE AND 5 INVERTEBRATE SPECIES [J].
NIELSEN, M ;
BRAESTRUP, C ;
SQUIRES, RF .
BRAIN RESEARCH, 1978, 141 (02) :342-346
[39]   SOME PROPERTIES OF DIAZEPAM-H-3 DISPLACING ACTIVITY FROM HUMAN-URINE [J].
NIELSEN, M ;
GREDAL, O ;
BRAESTRUP, C .
LIFE SCIENCES, 1979, 25 (08) :679-686
[40]  
NIELSEN M, BIOL PSYCHIATRY