THE ACTIVATION GATE OF THE SODIUM-CHANNEL CONTROLS BLOCKADE AND DEBLOCKADE BY DISOPYRAMIDE IN RABBIT PURKINJE-FIBERS

被引:22
作者
GRUBER, R [1 ]
CARMELIET, E [1 ]
机构
[1] LAB FYSIOL,B-3000 LEUVEN,BELGIUM
关键词
D O I
10.1111/j.1476-5381.1989.tb11921.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:41 / 50
页数:10
相关论文
共 27 条
[13]   ANTIARRHYTHMIC AGENTS - THE MODULATED RECEPTOR MECHANISM OF ACTION OF SODIUM AND CALCIUM CHANNEL-BLOCKING DRUGS [J].
HONDEGHEM, LM ;
KATZUNG, BG .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1984, 24 :387-423
[14]   TIME-DEPENDENT AND VOLTAGE-DEPENDENT INTERACTIONS OF ANTIARRHYTHMIC DRUGS WITH CARDIAC SODIUM CHANNELS [J].
HONDEGHEM, LM ;
KATZUNG, BG .
BIOCHIMICA ET BIOPHYSICA ACTA, 1977, 472 (3-4) :373-398
[15]   EFFECTS OF DISOPYRAMIDE ON THE MAXIMUM RATE OF RISE OF ACTION-POTENTIAL (VMAX) IN GUINEA-PIG PAPILLARY-MUSCLES [J].
KOJIMA, M ;
BAN, T ;
SADA, H .
JAPANESE JOURNAL OF PHARMACOLOGY, 1982, 32 (01) :91-102
[16]   DISOPYRAMIDE PHOSPHATE - IS IT JUST ANOTHER QUINIDINE [J].
KUS, T ;
SASYNIUK, BI .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1978, 56 (02) :326-331
[17]   SLOW RECOVERY OF THE MAXIMAL RATE OF RISE (VMAX) OF THE ACTION-POTENTIAL IN SHEEP CARDIAC PURKINJE-FIBERS [J].
SAIKAWA, T ;
CARMELIET, E .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1982, 394 (01) :90-93
[18]   LOCAL-ANESTHETICS - EFFECT OF PH ON USE-DEPENDENT BLOCK OF SODIUM CHANNELS IN FROG MUSCLE [J].
SCHWARZ, W ;
PALADE, PT ;
HILLE, B .
BIOPHYSICAL JOURNAL, 1977, 20 (03) :343-368
[19]   MECHANISMS OF USE-DEPENDENT BLOCK OF SODIUM-CHANNELS IN EXCITABLE-MEMBRANES BY LOCAL-ANESTHETICS [J].
STARMER, CF ;
GRANT, AO ;
STRAUSS, HC .
BIOPHYSICAL JOURNAL, 1984, 46 (01) :15-27
[20]   A QUANTITATIVE DESCRIPTION OF QX222-BLOCKADE OF SODIUM-CHANNELS IN SQUID AXONS [J].
STARMER, CF ;
YEH, JZ ;
TANGUY, J .
BIOPHYSICAL JOURNAL, 1986, 49 (04) :913-920