THE STRUCTURE OF A SYNTHETIC PEPSIN INHIBITOR COMPLEXED WITH ENDOTHIAPEPSIN

被引:54
作者
COOPER, J
FOUNDLING, S
HEMMINGS, A
BLUNDELL, T
JONES, DM
HALLETT, A
SZELKE, M
机构
[1] UNIV LONDON BIRKBECK COLL, DEPT CRYSTALLOG, MOLEC BIOL LAB, MALET ST, LONDON WC1E 7HX, ENGLAND
[2] ROYAL POSTGRAD MED SCH, DEPT CHEM PATHOL, LONDON W12 0HS, ENGLAND
来源
EUROPEAN JOURNAL OF BIOCHEMISTRY | 1987年 / 169卷 / 01期
关键词
D O I
10.1111/j.1432-1033.1987.tb13600.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:215 / 221
页数:7
相关论文
共 37 条
[1]  
ALBER T, 1983, CIBA F SYMP, V93, P4
[2]  
ANDREEVA NS, 1984, J BIOL CHEM, V259, P1353
[3]   MAPPING ACTIVE SITE OF PAPAIN WITH AID OF PEPTIDE SUBSTRATES AND INHIBITORS [J].
BERGER, A ;
SCHECHTER, I .
PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES, 1970, 257 (813) :249-+
[4]  
BLUNDELL TL, 1985, ASPARTIC PROTEINASES, P151
[5]   3-DIMENSIONAL STRUCTURE OF THE COMPLEX OF THE RHIZOPUS-CHINENSIS CARBOXYL PROTEINASE AND PEPSTATIN AT 2.5-A RESOLUTION [J].
BOTT, R ;
SUBRAMANIAN, E ;
DAVIES, DR .
BIOCHEMISTRY, 1982, 21 (26) :6956-6962
[6]   SPECIFIC-INHIBITION OF RENIN BY AN ANGIOTENSINOGEN ANALOG - STUDIES IN SODIUM DEPLETION AND RENIN-DEPENDENT HYPERTENSION [J].
BURTON, J ;
CODY, RJ ;
HERD, JA ;
HABER, E .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (09) :5476-5479
[7]   THE SYNTHESIS, PURIFICATION, AND EVALUATION OF A CHROMOPHORIC SUBSTRATE FOR PEPSIN AND OTHER ASPARTYL PROTEASES - DESIGN OF A SUBSTRATE BASED ON SUBSITE PREFERENCES [J].
DUNN, BM ;
KAMMERMANN, B ;
MCCURRY, KR .
ANALYTICAL BIOCHEMISTRY, 1984, 138 (01) :68-73
[8]   HIGH-RESOLUTION X-RAY ANALYSES OF RENIN INHIBITOR-ASPARTIC PROTEINASE COMPLEXES [J].
FOUNDLING, SI ;
COOPER, J ;
WATSON, FE ;
CLEASBY, A ;
PEARL, LH ;
SIBANDA, BL ;
HEMMINGS, A ;
WOOD, SP ;
BLUNDELL, TL ;
VALLER, MJ ;
NOREY, CG ;
KAY, J ;
BOGER, J ;
DUNN, BM ;
LECKIE, BJ ;
JONES, DM ;
ATRASH, B ;
HALLETT, A ;
SZELKE, M .
NATURE, 1987, 327 (6120) :349-352
[9]  
FRUTON JS, 1976, ADV ENZYMOL RAMB, V44, P1
[10]  
HALLETT A, 1985, ASPARTIC PROTEINASES, P467