DIFFERENCES IN RESULTS FROM INVIVO AND INVITRO STUDIES ON THE USE-DEPENDENCY OF N-METHYLASPARTATE ANTAGONISM BY MK-801 AND OTHER PHENCYCLIDINE RECEPTOR LIGANDS

被引:101
作者
DAVIES, SN [1 ]
MARTIN, D [1 ]
MILLAR, JD [1 ]
ARAM, JA [1 ]
CHURCH, J [1 ]
LODGE, D [1 ]
机构
[1] UNIV LONDON ROYAL VET COLL,DEPT PHYSIOL,ROYAL COLL ST,LONDON NW1 0TU,ENGLAND
关键词
D O I
10.1016/0014-2999(88)90225-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:141 / 151
页数:11
相关论文
共 21 条
[1]   THE DISSOCIATIVE ANESTHETICS, KETAMINE AND PHENCYCLIDINE, SELECTIVELY REDUCE EXCITATION OF CENTRAL MAMMALIAN NEURONS BY N-METHYL-ASPARTATE [J].
ANIS, NA ;
BERRY, SC ;
BURTON, NR ;
LODGE, D .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (02) :565-575
[2]  
ARAM J, 1986, British Journal of Pharmacology, V89, p778P
[3]  
ARAM JA, 1985, BR J PHARM, V86, pP539
[4]   COMPARISON OF SIGMA-OPIATE AND KAPPA-OPIATE RECEPTOR LIGANDS AS EXCITATORY AMINO-ACID ANTAGONISTS [J].
BERRY, SC ;
DAWKINS, SL ;
LODGE, D .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (01) :179-185
[5]  
CHURCH J, 1986, BR J PHARM, V90, pP10
[6]   MULTIPLE-CONDUCTANCE CHANNELS ACTIVATED BY EXCITATORY AMINO-ACIDS IN CEREBELLAR NEURONS [J].
CULLCANDY, SG ;
USOWICZ, MM .
NATURE, 1987, 325 (6104) :525-528
[7]  
FAGG GE, 1987, IN PRESS NEUROSCI LE
[8]   QUANTITATIVE STUDIES ON SOME ANTAGONISTS OF N-METHYL D-ASPARTATE IN SLICES OF RAT CEREBRAL-CORTEX [J].
HARRISON, NL ;
SIMMONDS, MA .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (02) :381-391
[9]   KETAMINE AND PHENCYCLIDINE CAUSE A VOLTAGE-DEPENDENT BLOCK OF RESPONSES TO L-ASPARTIC ACID [J].
HONEY, CR ;
MILJKOVIC, Z ;
MACDONALD, JF .
NEUROSCIENCE LETTERS, 1985, 61 (1-2) :135-139
[10]   GLUTAMATE ACTIVATES MULTIPLE SINGLE CHANNEL CONDUCTANCES IN HIPPOCAMPAL-NEURONS [J].
JAHR, CE ;
STEVENS, CF .
NATURE, 1987, 325 (6104) :522-525