SYNTHESIS OF 4-PHOSPHONO-DL-PHENYLALANINE AND OF 4-(PHOSPHONOMETHYL)-DL-PHENYLALANINE, 2 ANALOGS OF O-PHOSPHOTYROSINE

被引：25

作者：

BAYLELACOSTE, M

MOULINES, J

COLLIGNON, N

BOUMEKOUEZ, A

DETINGUYMOREAUD, E

NEUZIL, E

机构：

[1] INST NATL SCI APPL,IRCOF,COMPOSES ORGANOPHOSPHORES LAB,F-76131 MONT ST AIGNAN,FRANCE

[2] UNIV BORDEAUX 1,CHIM APPL LAB,F-33405 TALENCE,FRANCE

来源：

TETRAHEDRON | 1990年 / 46卷 / 23期

关键词：

D O I：

10.1016/S0040-4020(01)90076-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

:4-Phosphono-DL-phenylalanine 1 was synthetized from 4-bromo-DL-phenylalanine or from 4-(bromomethyl)-bromobenzene ; 4-(phosphonomethyl)-DL-phenylalanine 14 was prepared from methyl p-toluate. The interest of these phosphonic analogues arises from their possible interference in the metabolism of O-phosphotyrosine. © 1990.

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页码：7793 / 7802

页数：10

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