(-) BACLOFEN DECREASES NEUROTRANSMITTER RELEASE IN THE MAMMALIAN CNS BY AN ACTION AT A NOVEL GABA RECEPTOR

被引:953
作者
BOWERY, NG
HILL, DR
HUDSON, AL
DOBLE, A
MIDDLEMISS, DN
SHAW, J
TURNBULL, M
机构
[1] ICI LTD,DEPT BIOCHEM,ALDERLEY PK,CHESHIRE,ENGLAND
[2] ICI LTD,DEPT BIOL,ALDERLEY PK,CHESHIRE,ENGLAND
关键词
D O I
10.1038/283092a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:92 / 94
页数:3
相关论文
共 37 条
[1]  
ANDERSON SD, 1978, BRIT J PHARMACOL, V64, pP429
[2]  
ARBILLA S, 1978, BRIT J PHARMACOL, V63, pP389
[3]  
BOWERY NG, 1979, BRIT J PHARMACOL, V66, pP108
[4]  
BOWERY NG, 1979, BRIT J PHARMACOL, V67, pP444
[5]   DEPOLARIZING ACTIONS OF GAMMA-AMINOBUTYRIC ACID AND RELATED COMPOUNDS ON RAT SUPERIOR CERVICAL GANGLIA IN-VITRO [J].
BOWERY, NG ;
BROWN, DA .
BRITISH JOURNAL OF PHARMACOLOGY, 1974, 50 (02) :205-218
[6]  
BROWN DA, 1979, BRIT J PHARMACOL, V66, pP108
[7]   AXONAL GABA-RECEPTORS IN MAMMALIAN PERIPHERAL-NERVE TRUNKS [J].
BROWN, DA ;
MARSH, S .
BRAIN RESEARCH, 1978, 156 (01) :187-191
[8]   CENTRAL EFFECTS OF BETA-(PARA-CHLOROPHENYL)-GAMMA-AMINOBUTYRIC ACID [J].
CURTIS, DR ;
GAME, CJA ;
JOHNSTON, GA ;
MCCULLOCH, RM .
BRAIN RESEARCH, 1974, 70 (03) :493-499
[9]  
CURTIS DR, 1974, ERG PHYSIOL BIOL CH, V69, P97
[10]   BICUCULLINE, AN ANTAGONIST OF GABA AND SYNAPTIC INHIBITION IN SPINAL CORD OF CAT [J].
CURTIS, DR ;
DUGGAN, AW ;
FELIX, D ;
JOHNSTON, GA .
BRAIN RESEARCH, 1971, 32 (01) :69-&