ASSESSMENT OF NEUROLEPTIC POTENTIAL OF SOME NOVEL BENZAMIDE, BUTYROPHENONE, PHENOTHIAZINE AND INDOLE-DERIVATIVES

被引:28
作者
COSTALL, B [1 ]
FUNDERBURK, WH [1 ]
LEONARD, CA [1 ]
NAYLOR, RJ [1 ]
机构
[1] AH ROBINS CO,RES LABS,RICHMOND,VA 23220
关键词
D O I
10.1111/j.2042-7158.1978.tb13390.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:771 / 778
页数:8
相关论文
共 14 条
[1]   [1-[3-(PHENOTHIAZIN-10-YL)PROPYL]-4-PIPERIDINYL]PHENYLMETHANONES, A NOVEL CLASS OF LONG-ACTING NEUROLEPTIC AGENTS [J].
BOSWELL, RF ;
WELSTEAD, WJ ;
DUNCAN, RL ;
JOHNSON, DN ;
FUNDERBURK, WH .
JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (01) :136-139
[2]  
COSTALL B, 1973, ARZNEIMITTEL-FORSCH, V23, P674
[3]   COMPARISON OF ABILITIES OF TYPICAL NEUROLEPTIC AGENTS AND OF THIORIDAZINE, CLOZAPINE, SULPIRIDE AND METOCLOPRAMIDE TO ANTAGONIZE HYPERACTIVITY INDUCED BY DOPAMINE APPLIED INTRACEREBRALLY TO AREAS OF EXTRAPYRAMIDAL AND MESOLIMBIC SYSTEMS [J].
COSTALL, B ;
NAYLOR, RJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1976, 40 (01) :9-19
[4]   MESOLIMBIC INVOLVEMENT WITH BEHAVIORAL-EFFECTS INDICATING ANTIPSYCHOTIC ACTIVITY [J].
COSTALL, B ;
NAYLOR, RJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1974, 27 (01) :46-58
[5]  
COSTALL B, 1976, COCAINE OTHER STIMUL, P47
[6]  
DEGROOT J, 1959, VERH K NED AKAD WET, V52, P14
[7]   AROYLOPIPERIDINES AND PYRROLIDINES . A NEW CLASS OF POTENT CENTRAL NERVOUS SYSTEM DEPRESSANTS [J].
DUNCAN, RL ;
HELSLEY, GC ;
WELSTEAD, WJ ;
DAVANZO, JP ;
FUNDERBU.WH ;
LUNSFORD, CD .
JOURNAL OF MEDICINAL CHEMISTRY, 1970, 13 (01) :1-&
[8]   PSYCHOPHARMACOLOGICAL IMPLICATIONS OF DOPAMINE AND DOPAMINE ANTAGONISTS - CRITICAL EVALUATION OF CURRENT EVIDENCE [J].
HORNYKIEWICZ, O .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1977, 17 :545-559
[9]   COMPARISON OF INVITRO AND INVIVO DOPAMINE RECEPTOR ANTAGONISM PRODUCED BY SUBSTITUTED BENZAMIDE DRUGS [J].
JENNER, P ;
ELLIOTT, PNC ;
CLOW, A ;
REAVILL, C ;
MARSDEN, CD .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1978, 30 (01) :46-48
[10]   ANTAGONISM OF APOMORPHINE-INDUCED AND D-AMPHETAMINE-INDUCED STEREOTYPED BEHAVIOR BY INJECTION OF LOW-DOSES OF HALOPERIDOL INTO CAUDATE-NUCLEUS AND NUCLEUS ACCUMBENS [J].
PIJNENBURG, AJJ ;
HONIG, WMM ;
VANROSSUM, JM .
PSYCHOPHARMACOLOGIA, 1975, 45 (01) :65-71