TETRAMISOLE ANALOGS AS INHIBITORS OF ALKALINE-PHOSPHATASE, AN ENZYME INVOLVED IN RESISTANCE OF NEOPLASTIC-CELLS TO 6-THIOPURINES

被引：27

作者：

BHARGAVA, KK

LEE, MH

HUANG, YM

CUNNINGHAM, LS

AGRAWAL, KC

SARTORELLI, AC

机构：

[1] YALE UNIV,SCH MED,DEPT PHARMACOL,NEW HAVEN,CT 06510

[2] YALE UNIV,CTR COMPREHENS CANC,DEV THERAPEUT SECT,NEW HAVEN,CT 06510

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1977年 / 20卷 / 04期

关键词：

D O I：

10.1021/jm00214a021

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：563 / 566

页数：4

共 12 条

[1] CYTOCHEMICAL APPLICATION OF NEW POTENT INHIBITORS OF ALKALINE-PHOSPHATASES [J].

BORGERS, M .

JOURNAL OF HISTOCHEMISTRY & CYTOCHEMISTRY, 1973, 21 (09) :812-824

[2]

BORGERS M, 1975, HISTOCHEMISTRY, V44, P273

[3] NITROIMIDAZOLE DERIVATIVES . RELATIONSHIP BETWEEN STRUCTURE AND ANTITRICHOMONAL ACTIVITY [J].

BUTLER, K ;

HOWES, HL ;

LYNCH, JE ;

PIRIE, DK .

JOURNAL OF MEDICINAL CHEMISTRY, 1967, 10 (05) :891-&

[4] The synthesis of phenyl- and pyridyl-glyoxalines [J].

Clemo, GR ;

Holmes, T ;

Leith, GC .

JOURNAL OF THE CHEMICAL SOCIETY, 1938, :753-755

[5]

LEE MH, 1975, BIOCHEM PHARMACOL, V24, P1175

[6] SOLUBILIZATION AND PARTIAL-PURIFICATION OF ALKALINE-PHOSPHATASES OF SARCOMA 180/TG ASCITES-CELLS [J].

LEE, MH ;

SARTORELLI, AC .

BIOCHIMICA ET BIOPHYSICA ACTA, 1974, 358 (01) :69-81

[7] NOVEL BROAD-SPECTRUM ANTHELMINTICS . TETRAMISOLE AND RELATED DERIVATIVES OF 6-ARYLIMIDAZO[2,1-B)THIAZOLE [J].

RAEYMAEK.AH ;

ALLEWIJN, FT ;

VANDENBE.J ;

DEMOEN, PJA ;

VANOFFEN.TT ;

JANSSEN, PAJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1966, 9 (04) :545-+

[8]

ROSMAN M, 1974, CANCER RES, V34, P1952

[9]

SARTORELLI AC, 1975, PHARMACOL BASIS, P643

[10]

THIENPONT D, 1966, NATURE, V209, P1084

← 1 2 →