ANTIESTROGENS .2. STRUCTURE ACTIVITY STUDIES IN A SERIES OF 3-AROYL-2-ARYLBENZO[B]THIOPHENE DERIVATIVES LEADING TO [6-HYDROXY-2-(4-HYDROXYPHENYL)BENZO[B]THIEN-3-YL][4-[2-(1-PIPERIDINYL)ETHOXY]-PHENYL]METHANONE HYDROCHLORIDE (LY156758), A REMARKABLY EFFECTIVE ESTROGEN ANTAGONIST WITH ONLY MINIMAL INTRINSIC ESTROGENICITYO[

被引：273

作者：

JONES, CD

JEVNIKAR, MG

PIKE, AJ

PETERS, MK

BLACK, LJ

THOMPSON, AR

FALCONE, JF

CLEMENS, JA

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1984年 / 27卷 / 08期

关键词：

D O I：

10.1021/jm00374a021

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1057 / 1066

页数：10

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