DIFFERENTIAL-EFFECTS OF THE ENANTIOMERS OF 3-(3-HYDROXYPHENYL)-N-NORMAL-PROPYLPIPERIDINE (3-PPP) AT DOPAMINE RECEPTOR-SITES

被引:29
作者
KOCH, SW
KOE, BK
BACOPOULOS, NG
机构
[1] PFIZER INC,DIV CENT RES,DEPT METAB DIS & GEN PHARMACOL,GROTON,CT 06340
[2] DARTMOUTH COLL,HITCHCOCK MED CTR,DARTMOUTH MED SCH,DEPT PHARMACOL,HANOVER,NH 03755
[3] DARTMOUTH COLL,HITCHCOCK MED CTR,DARTMOUTH MED SCH,DEPT PSYCHIAT,HANOVER,NH 03755
关键词
D O I
10.1016/0014-2999(83)90299-6
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:279 / 283
页数:5
相关论文
共 10 条
[1]  
ARNT J, 1983, European Journal of Pharmacology, V86, P185
[2]   DOPAMINE-RECEPTORS IN RAT-BRAIN REGIONS - OPTIMAL CONDITIONS FOR H-3-AGONIST BINDING, PH DEPENDENCY AND LACK OF INHIBITION BY ASCORBIC-ACID [J].
BACOPOULOS, NG .
BIOCHEMICAL PHARMACOLOGY, 1982, 31 (19) :3085-3091
[3]  
CLEMENTCORMIER YC, 1974, P NAT ACAD SCI US, V71, P1112
[4]   3-PPP, A NEW CENTRALLY ACTING DA-RECEPTOR AGONIST WITH SELECTIVITY FOR AUTORECEPTORS [J].
HJORTH, S ;
CARLSSON, A ;
WIKSTROM, H ;
LINDBERG, P ;
SANCHEZ, D ;
HACKSELL, U ;
ARVIDSSON, LE ;
SVENSSON, U ;
NILSSON, JLG .
LIFE SCIENCES, 1981, 28 (11) :1225-1238
[5]   PHARMACOLOGICAL PROFILES OF THE PUTATIVE DOPAMINE AUTORECEPTOR AGONISTS 3-PPP AND TL-99 [J].
MARTIN, GE ;
HAUBRICH, DR ;
WILLIAMS, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 76 (01) :15-23
[6]  
MELTZER LT, 1982, SOC NEUR ABSTR, V8, P922
[7]  
PATRICK RL, 1981, J PHARM EXP THER, V217, P868
[8]  
ROTH RH, 1979, COMMUN PSYCHOPHARMAC, V3, P429
[9]  
WAGGONER WG, 1980, MOL PHARMACOL, V18, P91
[10]   INHIBITION OF POSTSYNAPTIC DOPAMINE-SENSITIVE ADENYLATE-CYCLASE IN CARP RETINA BY THE PUTATIVE DOPAMINE AUTORECEPTOR AGONIST, 3-PPP [J].
WATLING, KJ ;
JONES, JH ;
WILLIAMS, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 82 (1-2) :117-118