RATIONALE FOR DESIGN OF BIOLOGICALLY REVERSIBLE DRUG DERIVATIVES - PRODRUGS

被引:226
作者
SINKULA, AA [1 ]
YALKOWSKY, SH [1 ]
机构
[1] UPJOHN CO, RES LABS, KALAMAZOO, MI 49001 USA
关键词
D O I
10.1002/jps.2600640203
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:181 / 210
页数:30
相关论文
共 419 条
[1]   PROPERTIES OF THE ACID PHOSPHATASES OF ERYTHROCYTES AND OF THE HUMAN PROSTATE GLAND [J].
ABULFADL, MAM ;
KING, EJ .
BIOCHEMICAL JOURNAL, 1949, 45 (01) :51-60
[2]  
AKERMAN B, 1966, ACTA PHARMACOL TOX, V24, P389
[3]  
AKERMAN SBA, 1973, ACTA PHARMACOL TOX, V32, P88
[4]  
ALBERT A, 1960, SELECTIVE TOXICITY, P30
[5]  
ALBERT A, 1964, SELECTIVE TOXICITY, P57
[7]  
Alles GA, 1940, J BIOL CHEM, V133, P375
[8]  
ALTMAN PA, 1964, BIOLOGY DATA BOOK, P279
[9]   SOLUBILITY OF NONELECTROLYTES IN POLAR-SOLVENTS .2. SOLUBILITY OF ALIPHATIC-ALCOHOLS IN WATER [J].
AMIDON, GL ;
YALKOWSKY, SH ;
LEUNG, S .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1974, 63 (12) :1858-1866
[10]  
AMOORE JE, 1970, J SOC COSMET CHEM, V21, P99