SPECIFIC BINDING OF [H-3]LABELED NITRENDIPINE TO MEMBRANES FROM CORONARY-ARTERIES AND HEART IN RELATION TO PHARMACOLOGICAL EFFECTS - PARADOXICAL STIMULATION BY DILTIAZEM

被引:180
作者
DEPOVER, A
MATLIB, MA
LEE, SW
DUBE, GP
GRUPP, IL
GRUPP, G
SCHWARTZ, A
机构
[1] UNIV CINCINNATI,COLL MED,DEPT PHARMACOL,CINCINNATI,OH 45267
[2] UNIV CINCINNATI,COLL MED,DEPT CELL BIOPHYS,CINCINNATI,OH 45267
[3] UNIV CINCINNATI,COLL MED,DEPT PHYSIOL,CINCINNATI,OH 45267
[4] UNIV CINCINNATI,COLL MED,DEPT MED,DIV CARDIOL,CINCINNATI,OH 45267
关键词
D O I
10.1016/0006-291X(82)91838-1
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:110 / 117
页数:8
相关论文
共 17 条
[1]  
BELLEMANN P, 1981, ARZNEIMITTEL-FORSCH, V31-2, P2064
[2]   HIGH-AFFINITY BINDING OF A CALCIUM-CHANNEL ANTAGONIST TO SMOOTH AND CARDIAC-MUSCLE [J].
BOLGER, GT ;
GENGO, PJ ;
LUCHOWSKI, EM ;
SIEGEL, H ;
TRIGGLE, DJ ;
JANIS, RA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 104 (04) :1604-1609
[3]   EFFECT OF SULOCTIDIL ON NA+-K+ ATPASE ACTIVITY AND ON MEMBRANE FLUIDITY IN RAT-BRAIN SYNAPTOSOMES [J].
CHATELAIN, P ;
RECKINGER, N ;
RONCUCCI, R .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (24) :3677-3680
[4]   THE INTERACTION OF [H-3]-LABELED NITRENDIPINE WITH RECEPTORS FOR CALCIUM-ANTAGONISTS IN THE CEREBRAL-CORTEX AND HEART OF RATS [J].
EHLERT, FJ ;
ITOGA, E ;
ROESKE, WR ;
YAMAMURA, HI .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 104 (03) :937-943
[5]   THE BINDING OF [H-3]-LABELED NITRENDIPINE TO RECEPTORS FOR CALCIUM-CHANNEL ANTAGONISTS IN THE HEART, CEREBRAL-CORTEX, AND ILEUM OF RATS [J].
EHLERT, FJ ;
ROESKE, WR ;
ITOGA, E ;
YAMAMURA, HI .
LIFE SCIENCES, 1982, 30 (25) :2191-2202
[6]   SPECIFIC PHARMACOLOGY OF CALCIUM IN MYOCARDIUM, CARDIAC-PACEMAKERS, AND VASCULAR SMOOTH-MUSCLE [J].
FLECKENSTEIN, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1977, 17 :149-166
[7]   BLOCKADE OR REVERSAL OF CONTRACTION INDUCED BY CALCIUM AND ADRENALINE IN DEPOLARIZED ARTERIAL SMOOTH MUSCLE [J].
GODFRAIND, T ;
KABA, A .
BRITISH JOURNAL OF PHARMACOLOGY, 1969, 36 (03) :549-+
[8]  
GRUPP G, 1982, J PHARMACOL EXP THER, V220, P145
[9]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265
[10]  
MATLIB MA, 1979, J BIOL CHEM, V254, P1834