CGS-8216 - RECEPTOR-BINDING CHARACTERISTICS OF A POTENT BENZODIAZEPINE ANTAGONIST

被引:206
作者
CZERNIK, AJ
PETRACK, B
KALINSKY, HJ
PSYCHOYOS, S
CASH, WD
TSAI, C
RINEHART, RK
GRANAT, FR
LOVELL, RA
BRUNDISH, DE
WADE, R
机构
[1] CIBA GEIGY CORP, SUMMIT, NJ 07901 USA
[2] CIBA GEIGY, DIV PHARMACEUT, RES CTR, HORSHAM, W SUSSEX, ENGLAND
关键词
D O I
10.1016/0024-3205(82)90573-2
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:363 / 372
页数:10
相关论文
共 22 条
[1]  
BENNETT JP, 1978, NEUROTRANSMITTER REC, P57
[2]   BRAIN SPECIFIC BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SQUIRES, RF .
BRITISH JOURNAL OF PSYCHIATRY, 1978, 133 (SEP) :249-260
[3]   SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].
BRAESTRUP, C ;
SQUIRES, RF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809
[4]  
BRUNS RF, 1980, CAN J PHYSIOL PHARM, V58, P673, DOI 10.1139/y80-110
[5]   BENZODIAZEPINE RECEPTORS - LABELING IN INTACT ANIMALS WITH [H-3]FLUNITRAZEPAM [J].
CHANG, RSL ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (02) :213-218
[6]   PREPARATION AND PROPERTIES OF A CELL-FREE HORMONALLY RESPONSIVE ADENYLATE CYCLASE FROM GUINEA-PIG BRAIN [J].
CHASIN, M ;
MAMRAK, F ;
SAMANIEGO, SG .
JOURNAL OF NEUROCHEMISTRY, 1974, 22 (06) :1031-1038
[7]  
CHASIN M, 1972, METHODS CYCLIC NUCLE, P176
[8]  
EHLERT FJ, 1981, LIFE SCI, V29, P235, DOI 10.1016/0024-3205(81)90239-3
[9]   SELECTIVE ANTAGONISTS OF BENZODIAZEPINES [J].
HUNKELER, W ;
MOHLER, H ;
PIERI, L ;
POLC, P ;
BONETTI, EP ;
CUMIN, R ;
SCHAFFNER, R ;
HAEFELY, W .
NATURE, 1981, 290 (5806) :514-516
[10]   RESOLUTION OF 2 BIOCHEMICALLY AND PHARMACOLOGICALLY DISTINCT BENZODIAZEPINE RECEPTORS [J].
KLEPNER, CA ;
LIPPA, AS ;
BENSON, DI ;
SANO, MC ;
BEER, B .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1979, 11 (04) :457-462