ANION-DEPENDENT MODULATION OF [H-3]MUSCIMOL BINDING AND OF GABA-STIMULATED [H-3-LABELED FLUNITRAZEPAM BINDING BY PICROTOXIN AND RELATED CNS CONVULSANTS

被引：29

作者：

SUPAVILAI, P

MANNONEN, A

COLLINS, JF

KAROBATH, M

机构：

[1] SANDOZ LTD,PRECLIN RES,CH-4002 BASEL,SWITZERLAND

[2] CITY LONDON POLYTECH,DEPT CHEM,LONDON EC3N 2EY,ENGLAND

来源：

EUROPEAN JOURNAL OF PHARMACOLOGY | 1982年 / 81卷 / 04期

关键词：

D O I：

10.1016/0014-2999(82)90362-4

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：687 / 691

页数：5

共 13 条

[1] MUSCIMOL BINDING IN RAT-BRAIN - ASSOCIATION WITH SYNAPTIC GABA RECEPTORS [J].

BEAUMONT, K ;

CHILTON, WS ;

YAMAMURA, HI ;

ENNA, SJ .

BRAIN RESEARCH, 1978, 148 (01) :153-162

[2]

BOWERY NG, 1976, NATURE, V261, P5561

[3] STEREOSPECIFICITY AND STRUCTURE-ACTIVITY REQUIREMENTS OF GABA RECEPTOR-BINDING IN RAT-BRAIN [J].

ENNA, SJ ;

COLLINS, JF ;

SNYDER, SH .

BRAIN RESEARCH, 1977, 124 (01) :185-190

[4] A STEROID DERIVATIVE, R-5135, ANTAGONIZES THE GABA-BENZODIAZEPINE RECEPTOR INTERACTION [J].

HUNT, P ;

CLEMENTSJEWERY, S .

NEUROPHARMACOLOGY, 1981, 20 (04) :357-361

[5] STRUCTURAL ASPECTS OF PICROTOXININ ACTION [J].

JARBOE, CH ;

PORTER, LA ;

BUCKLER, RT .

JOURNAL OF MEDICINAL CHEMISTRY, 1968, 11 (04) :729-&

[6] MODULATION BY PICROTOXIN AND IPTBO OF FLUNITRAZEPAM-H-3 BINDING TO THE GABA-BENZODIAZEPINE RECEPTOR COMPLEX OF RAT CEREBELLUM [J].

KAROBATH, M ;

DREXLER, G ;

SUPAVILAI, P .

LIFE SCIENCES, 1981, 28 (03) :307-313

[7]

KUBO Y, 1981, NEUROSCI LETT, V25, P83

[8]

LEBEDA FJ, 1981, SOC NEUROSCI ABSTR, V7, P124

[9] THE INHIBITION OF GABA-STIMULATED BENZODIAZEPINE BINDING BY A CONVULSANT BENZODIAZEPINE [J].

OBRIEN, RA ;

SPIRT, NM .

LIFE SCIENCES, 1980, 26 (17) :1441-1445

[10] PICROTOXIN AND CONVULSANT BINDING-SITES IN MAMMALIAN BRAIN [J].

OLSEN, RW ;

LEEBLUNDBERG, F ;

NAPIAS, C .

BRAIN RESEARCH BULLETIN, 1980, 5 :217-221

← 1 2 →