1,3-DIALKYL-8-(PARA-SULFOPHENYL)XANTHINES - POTENT WATER-SOLUBLE ANTAGONISTS FOR A1-ADENOSINE AND A2-ADENOSINE RECEPTORS

被引：273

作者：

DALY, JW

PADGETT, W

SHAMIM, MT

BUTTSLAMB, P

WATERS, J

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 04期

关键词：

D O I：

10.1021/jm00382a018

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：487 / 492

页数：6

共 34 条

[1] 8-ARYLTHEOPHYLLINES [J].

BARIANA, DS .

CANADIAN JOURNAL OF CHEMISTRY, 1968, 46 (21) :3413-&

[2] REACTIONS OF 1,3-DIMETHYL-5,6-DIAMINOURACIL [J].

BLICKE, FF ;

GODT, HC .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1954, 76 (10) :2798-2800

[3] ADENOSINE RECEPTOR-BINDING - STRUCTURE-ACTIVITY ANALYSIS GENERATES EXTREMELY POTENT XANTHINE ANTAGONISTS [J].

BRUNS, RF ;

DALY, JW ;

SNYDER, SH .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (07) :2077-2080

[4] ADENOSINE ANTAGONISM BY PURINES, PTERIDINES AND BENZOPTERIDINES IN HUMAN-FIBROBLASTS [J].

BRUNS, RF .

BIOCHEMICAL PHARMACOLOGY, 1981, 30 (04) :325-333

[5]

BRUNS RF, 1980, CAN J PHYSIOL PHARM, V58, P673, DOI 10.1139/y80-110

[6] ADENOSINE RECEPTORS IN BRAIN MEMBRANES - BINDING OF N6-CYCLOHEXYL[H-3]ADENOSINE AND 1,3-DIETHYL-8-[H-3]PHENYLXANTHINE [J].

BRUNS, RF ;

DALY, JW ;

SNYDER, SH .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (09) :5547-5551

[7] ADENOSINE RECEPTORS IN THE CENTRAL NERVOUS-SYSTEM - RELATIONSHIP TO THE CENTRAL ACTIONS OF METHYLXANTHINES [J].

DALY, JW ;

BRUNS, RF ;

SNYDER, SH .

LIFE SCIENCES, 1981, 28 (19) :2083-2097

[8] ADENOSINE RECEPTORS - TARGETS FOR FUTURE DRUGS [J].

DALY, JW .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (03) :197-207

[9]

DALY JW, 1983, CELL MOL NEUROBIOL, V3, P6

[10]

FIESER LF, 1977, REAGENTS ORGANIC SYN, V1, P1180

← 1 2 3 4 →