BETA-1-SELECTIVE ADRENOCEPTOR ANTAGONISTS .1. SYNTHESIS AND BETA-ADRENERGIC BLOCKING ACTIVITY OF A SERIES OF BINARY (ARYLOXY)PROPANOLAMINES

被引：81

作者：

KIERSTEAD, RW

FARAONE, A

MENNONA, F

MULLIN, J

GUTHRIE, RW

CROWLEY, H

SIMKO, B

BLABER, LC

机构：

[1] HOFFMANN LA ROCHE INC, DEPT PHARMACOL, NUTLEY, NJ 07110 USA

[2] ROCHE PROD LTD, DEPT PHARMACOL, WELWYN GARDEN CITY AL7 3AY, HERTS, ENGLAND

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1983年 / 26卷 / 11期

关键词：

D O I：

10.1021/jm00365a004

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1561 / 1569

页数：9

共 13 条

[1]

BAER E, 1952, BIOCHEM PREPARAT, V2, P31

[2]

CASTANER J, 1979, DRUGS FUTURE, V4, P46

[3]

CASTILLO JC, 1947, J PHARMACOL EXP THER, V90, P104

[4]

COMER WT, 1979, MED CHEM 2, P1050

[5]

FAHRENHOLTZ KE, 1980, Patent No. 4202979

[6] REDUCTIVE CLEAVAGE OF SULFONAMIDES WITH SODIUM BIS(2-METHOXYETHOXY)ALUMINUM HYDRIDE [J].

GOLD, EH ;

BABAD, E .

JOURNAL OF ORGANIC CHEMISTRY, 1972, 37 (13) :2208-&

[7] STUDIES IN PROSTAGLANDINS .10. SYNTHESIS OF PROSTAGLANDIN MODELS AND PROSTAGLANDINS BY CONJUGATE ADDITION OF A FUNCTIONALIZED ORGANOCOPPER REAGENT [J].

KLUGE, AF ;

UNTCH, KG ;

FRIED, JH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1972, 94 (22) :7827-&

[8] BETA-1-SELECTIVE ADRENOCEPTOR ANTAGONISTS .2. 4-ETHER-LINKED PHENOXYPROPANOLAMINES [J].

MACHIN, PJ ;

HURST, DN ;

BRADSHAW, RM ;

BLABER, LC ;

BURDEN, DT ;

FRYER, AD ;

MELARANGE, RA ;

SHIVDASANI, C .

JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (11) :1570-1576

[9] CONVERSION OF 1,2-DIOLS VIA CYCLIC ORTHO ACETATES TO ACETATES OF CHLOROHYDRINS BY TREATMENT WITH TRIMETHYLSILYL CHLORIDE [J].

NEWMAN, MS ;

OLSON, DR .

JOURNAL OF ORGANIC CHEMISTRY, 1973, 38 (24) :4203-4204

[10]

ULRICH H, 1962, Patent No. 1138314

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