DUAL EFFECT OF N-ETHYLMALEIMIDE ON AGONIST-MEDIATED CONFORMATIONAL-CHANGES OF BETA-ADRENERGIC RECEPTORS

被引:20
作者
ANDRE, C [1 ]
VAUQUELIN, G [1 ]
SEVERNE, Y [1 ]
DEBACKER, JP [1 ]
STROSBERG, AD [1 ]
机构
[1] UNIV PARIS 07,CNRS,IRBM,IMMUNOL MOLEC LAB,F-75221 PARIS 05,FRANCE
关键词
D O I
10.1016/0006-2952(82)90591-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3657 / 3662
页数:6
相关论文
共 17 条
[1]  
BIRD SJ, 1978, J BIOL CHEM, V253, P8826
[2]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[3]   TISSUE SULFHYDRYL GROUPS [J].
ELLMAN, GL .
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1959, 82 (01) :70-77
[4]  
HOWLETT AC, 1978, MOL PHARMACOL, V14, P531
[5]   DISTINCTION BETWEEN 2 SUB-POPULATIONS OF BETA-1-ADRENERGIC RECEPTORS IN HUMAN ADIPOSE-CELLS [J].
JACOBSSON, B ;
VAUQUELIN, G ;
WESSLAU, C ;
SMITH, U ;
STROSBERG, AD .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1981, 114 (02) :349-354
[6]  
JEFFERY DR, 1980, J BIOL CHEM, V255, P5015
[7]  
KENT RS, 1980, MOL PHARMACOL, V17, P14
[8]  
LAD PM, 1980, J BIOL CHEM, V255, P988
[9]   AGONIST-PROMOTED COUPLING OF THE BETA-ADRENERGIC-RECEPTOR WITH THE GUANINE-NUCLEOTIDE REGULATORY PROTEIN OF THE ADENYLATE-CYCLASE SYSTEM [J].
LIMBIRD, LE ;
GILL, DM ;
LEFKOWITZ, RJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (02) :775-779
[10]  
STADEL JM, 1979, MOL PHARMACOL, V16, P709