QUANTITATIVE AUTORADIOGRAPHY OF [H-3]-MK-801 BINDING-SITES IN MAMMALIAN BRAIN

被引:171
作者
BOWERY, NG [1 ]
WONG, EHF [1 ]
HUDSON, AL [1 ]
机构
[1] MERCK SHARP & DOHME RES LABS, NEUROSCI RES CTR, HARLOW CM20 2QR, ESSEX, ENGLAND
关键词
D O I
10.1111/j.1476-5381.1988.tb11484.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:944 / 954
页数:11
相关论文
共 41 条
[1]   THE DISSOCIATIVE ANESTHETICS, KETAMINE AND PHENCYCLIDINE, SELECTIVELY REDUCE EXCITATION OF CENTRAL MAMMALIAN NEURONS BY N-METHYL-ASPARTATE [J].
ANIS, NA ;
BERRY, SC ;
BURTON, NR ;
LODGE, D .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (02) :565-575
[2]  
BENEVIDES J, 1987, BRIT J PHARMACOL, V90, pP280
[3]  
BOWERY N G, 1986, British Journal of Pharmacology, V89, p775P
[4]  
BOWERY NG, 1987, 10TH P IUPHAR C SYDN
[5]  
Chang Y., 1973, BIOCHEM PHARMACOL, V22, P3099
[6]   ANTICONVULSANT ACTIVITY OF (+)-5-METHYL-10, 11-DIHYDRO-5H-DIBENZO[A,D]CYCLOHEPTEN-5, 10-IMINE (MK-801), A SUBSTANCE WITH POTENT ANTICONVULSANT, CENTRAL SYMPATHOMIMETIC, AND APPARENT ANXIOLYTIC PROPERTIES [J].
CLINESCHMIDT, BV ;
MARTIN, GE ;
BUNTING, PR .
DRUG DEVELOPMENT RESEARCH, 1982, 2 (02) :123-134
[7]   AUTORADIOGRAPHIC DISTRIBUTION OF PHENCYCLIDINE RECEPTORS IN THE RAT-BRAIN USING [3H]1-(1-(2-THIENYL)CYCLOHEXYL)PIPERIDINE([3H]TCP) [J].
CONTRERAS, PC ;
QUIRION, R ;
ODONOHUE, TL .
NEUROSCIENCE LETTERS, 1986, 67 (02) :101-106
[8]   THE EFFECTS OF A SERIES OF OMEGA-PHOSPHONIC ALPHA-CARBOXYLIC AMINO-ACIDS ON ELECTRICALLY EVOKED AND EXCITANT AMINO ACID-INDUCED RESPONSES IN ISOLATED SPINAL-CORD PREPARATIONS [J].
EVANS, RH ;
FRANCIS, AA ;
JONES, AW ;
SMITH, DAS ;
WATKINS, JC .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 75 (01) :65-75
[9]   PHENCYCLIDINE AND RELATED DRUGS BIND TO THE ACTIVATED N-METHYL-D-ASPARTATE RECEPTOR CHANNEL COMPLEX IN RAT-BRAIN MEMBRANES [J].
FAGG, GE .
NEUROSCIENCE LETTERS, 1987, 76 (02) :221-227
[10]   EXCITATORY AMINO-ACID SYNAPTIC MECHANISMS AND NEUROLOGICAL FUNCTION [J].
FAGG, GE ;
FOSTER, AC ;
GANONG, AH .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1986, 7 (09) :357-363