RELATIVE AFFINITIES OF DRUGS ACTING AT CHOLINOCEPTORS IN DISPLACING AGONIST AND ANTAGONIST RADIOLIGANDS - THE NMS OXO-M RATIO AS AN INDEX OF EFFICACY AT CORTICAL MUSCARINIC RECEPTORS

被引:131
作者
FREEDMAN, SB
HARLEY, EA
IVERSEN, LL
机构
关键词
D O I
10.1111/j.1476-5381.1988.tb11451.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:437 / 445
页数:9
相关论文
共 32 条
[1]   CHARACTER OF THE MUSCARINIC RECEPTORS IN DIFFERENT REGIONS OF THE RAT-BRAIN [J].
BIRDSALL, NJM ;
HULME, EC ;
BURGEN, A .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1980, 207 (1166) :1-12
[2]  
BIRDSALL NJM, 1978, MOL PHARMACOL, V14, P723
[3]  
BIRDSALL NJM, 1986, ADV BEHAVIOURAL BIOL, V29, P565
[4]   INOSITOL PHOSPHOLIPID HYDROLYSIS IN RAT CEREBRAL CORTICAL SLICES .1. RECEPTOR CHARACTERIZATION [J].
BROWN, E ;
KENDALL, DA ;
NAHORSKI, SR .
JOURNAL OF NEUROCHEMISTRY, 1984, 42 (05) :1379-1387
[5]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[6]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[7]  
EGLEN RM, 1986, J AUTON PHARMACOL, V5, P323
[8]  
EHLERT FJ, 1985, MOL PHARMACOL, V28, P410
[9]   GUANINE-NUCLEOTIDE REGULATION OF AGONIST BINDING TO MUSCARINIC CHOLINERGIC RECEPTORS - RELATION TO EFFICACY OF AGONISTS FOR STIMULATION OF PHOSPHOINOSITIDE BREAKDOWN AND CA-2+ MOBILIZATION [J].
EVANS, T ;
HEPLER, JR ;
MASTERS, SB ;
BROWN, JH ;
HARDEN, TK .
BIOCHEMICAL JOURNAL, 1985, 232 (03) :751-757
[10]   NEW PROBE FOR HETEROGENEITY IN MUSCARINIC RECEPTORS - 2-METHYL-SPIRO-(1,3-DIOXOLANE-4,3')-QUINUCLIDINE [J].
FISHER, A ;
WEINSTOCK, M ;
GITTER, S ;
COHEN, S .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1976, 37 (02) :329-338