SELECTIVITIES OF OPIOID PEPTIDE ANALOGS AS AGONISTS AND ANTAGONISTS AT THE DELTA-RECEPTOR

被引：187

作者：

CORBETT, AD

GILLAN, MGC

KOSTERLITZ, HW

MCKNIGHT, AT

PATERSON, SJ

ROBSON, LE

机构：

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 1984年 / 83卷 / 01期

关键词：

D O I：

10.1111/j.1476-5381.1984.tb10143.x

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：271 / 279

页数：9

共 17 条

[1] DYNORPHIN1-8 AND DYNORPHIN1-9 ARE LIGANDS FOR THE KAPPA-SUBTYPE OF OPIATE RECEPTOR [J].

CORBETT, AD ;

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MAGNAN, J ;

KOSTERLITZ, HW .

NATURE, 1982, 299 (5878) :79-81

[2] ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR [J].

COTTON, R ;

GILES, MG ;

MILLER, L ;

SHAW, JS ;

TIMMS, D .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 97 (3-4) :331-332

[3] [H-3]TYR-D-SER-GLY-PHE-LEU-THR - A SPECIFIC PROBE FOR THE DELTA-OPIATE RECEPTOR SUBTYPE IN BRAIN MEMBRANES [J].

DAVID, M ;

MOISAND, C ;

MEUNIER, JC ;

MORGAT, JL ;

GACEL, G ;

ROQUES, BP .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 78 (03) :385-387

[4] TYR-D-SER-GLY-PHE-LEU-THR, A HIGHLY PREFERENTIAL LIGAND FOR DELTA-OPIATE RECEPTORS [J].

GACEI, G ;

FOURNIEZALUSKI, MC ;

ROQUES, BP .

FEBS LETTERS, 1980, 118 (02) :245-247

[5] SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN [J].

GILLAN, MGC ;

KOSTERLITZ, HW .

BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (03) :461-468

[6] EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS [J].

HUGHES, J ;

KOSTERLITZ, HW ;

LESLIE, FM .

BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :371-381

[7] ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS [J].

LORD, JAH ;

WATERFIELD, AA ;

HUGHES, J ;

KOSTERLITZ, HW .

NATURE, 1977, 267 (5611) :495-499

[8] THE BINDING SPECTRUM OF NARCOTIC ANALGESIC DRUGS WITH DIFFERENT AGONIST AND ANTAGONIST PROPERTIES [J].

MAGNAN, J ;

PATERSON, SJ ;

TAVANI, A ;

KOSTERLITZ, HW .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 319 (03) :197-205

[9] INCREASE IN POTENCIES OF OPIOID-PEPTIDES AFTER PEPTIDASE INHIBITION [J].

MCKNIGHT, AT ;

CORBETT, AD ;

KOSTERLITZ, HW .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 86 (3-4) :393-402

[10] BIS-PENICILLAMINE ENKEPHALINS POSSESS HIGHLY IMPROVED SPECIFICITY TOWARD DELTA-OPIOID RECEPTORS [J].

MOSBERG, HI ;

HURST, R ;

HRUBY, VJ ;

GEE, K ;

YAMAMURA, HI ;

GALLIGAN, JJ ;

BURKS, TF .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (19) :5871-5874

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