BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF [H-3] GBR-12935 BINDING INVITRO TO RAT STRIATAL MEMBRANES - LABELING OF THE DOPAMINE UPTAKE COMPLEX

被引:271
作者
ANDERSEN, PH
机构
关键词
D O I
10.1111/j.1471-4159.1987.tb05752.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
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页码:1887 / 1896
页数:10
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共 30 条
[1]   [H-3] GBR-12935 - A SPECIFIC HIGH-AFFINITY LIGAND FOR LABELING THE DOPAMINE TRANSPORT COMPLEX [J].
BERGER, P ;
JANOWSKY, A ;
VOCCI, F ;
SKOLNICK, P ;
SCHWERI, MM ;
PAUL, SM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 107 (02) :289-290
[2]   HIGH-AFFINITY [H-3] GBR 12783 BINDING TO A SPECIFIC SITE ASSOCIATED WITH THE NEURONAL DOPAMINE UPTAKE COMPLEX IN THE CENTRAL-NERVOUS-SYSTEM [J].
BONNET, JJ ;
PROTAIS, P ;
CHAGRAOUI, A ;
COSTENTIN, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) :211-222
[3]   GBR-12783, A POTENT AND SELECTIVE INHIBITOR OF DOPAMINE UPTAKE - BIOCHEMICAL-STUDIES INVIVO AND EXVIVO [J].
BONNET, JJ ;
COSTENTIN, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 121 (02) :199-209
[4]   SIMULTANEOUS EVALUATION BY A DOUBLE LABELING METHOD OF DRUG-INDUCED UPTAKE INHIBITION AND RELEASE OF DOPAMINE IN SYNAPTOSOMAL PREPARATION OF RAT STRIATUM [J].
BONNET, JJ ;
LEMASSON, MH ;
COSTENTIN, J .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (13) :2129-2135
[5]  
BURKARD WP, 1985, 1984 P S DICL, P1
[6]   BINDING CHARACTERISTICS OF THE DOPAMINE UPTAKE INHIBITOR [H-3] NOMIFENSINE TO STRIATAL MEMBRANES [J].
DUBOCOVICH, ML ;
ZAHNISER, NR .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (08) :1137-1144
[7]   BEHAVIORAL PROPERTIES OF GBR-12909, GBR-13069 AND GBR-13098 - SPECIFIC INHIBITORS OF DOPAMINE UPTAKE [J].
HEIKKILA, RE ;
MANZINO, L .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 103 (3-4) :241-248
[8]   EFFECTS OF 1-METHYL-4-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE AND RELATED-COMPOUNDS ON THE UPTAKE OF [H-3]3,4-DIHYDROXYPHENYLETHYLAMINE AND [H-3]5-HYDROXYTRYPTAMINE IN NEOSTRIATAL SYNAPTOSOMAL PREPARATIONS [J].
HEIKKILA, RE ;
YOUNGSTER, SK ;
MANZINO, L ;
CABBAT, FS ;
DUVOISIN, RC .
JOURNAL OF NEUROCHEMISTRY, 1985, 44 (01) :310-313
[9]   NEUROCHEMICAL PROFILE OF LU-19-005, A POTENT INHIBITOR OF UPTAKE OF DOPAMINE, NORADRENALINE, AND SEROTONIN [J].
HYTTEL, J ;
LARSEN, JJ .
JOURNAL OF NEUROCHEMISTRY, 1985, 44 (05) :1615-1622
[10]  
HYTTEL J, 1984, CRC HDB STEREOISOMER, P143