AN INHIBITOR OF PROTEIN-KINASE-C, 1-(5-ISOQUINOLINYLSULFONYL)-2-METHYLPIPERAZINE(H-7) INHIBITS TPA-INDUCED REDUCTION OF VINCRISTINE UPTAKE FROM P388 MURINE LEUKEMIC-CELL

被引:42
作者
IDO, M [1 ]
ASAO, T [1 ]
SAKURAI, M [1 ]
INAGAKI, M [1 ]
SAITO, M [1 ]
HIDAKA, H [1 ]
机构
[1] MIE UNIV,SCH MED,DEPT PEDIAT & PHARMACOL,TSU,MIE 514,JAPAN
关键词
D O I
10.1016/0145-2126(86)90050-0
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:1063 / 1069
页数:7
相关论文
共 23 条
[1]  
CHERVINSKY DS, 1976, J MED, V7, P63
[2]   ACTIVE OUTWARD TRANSPORT OF DAUNOMYCIN IN RESISTANT EHRLICH ASCITES TUMOR-CELLS [J].
DANO, K .
BIOCHIMICA ET BIOPHYSICA ACTA, 1973, 323 (03) :466-483
[3]  
HELFMAN DM, 1983, CANCER RES, V43, P2955
[4]   ISOQUINOLINESULFONAMIDES, NOVEL AND POTENT INHIBITORS OF CYCLIC-NUCLEOTIDE DEPENDENT PROTEIN-KINASE AND PROTEIN KINASE-C [J].
HIDAKA, H ;
INAGAKI, M ;
KAWAMOTO, S ;
SASAKI, Y .
BIOCHEMISTRY, 1984, 23 (21) :5036-5041
[5]   PHORBOL ESTER STIMULATION OF INSULIN RELEASE AND SECRETORY-GRANULE PROTEIN-PHOSPHORYLATION IN A TRANSPLANTABLE RAT INSULINOMA [J].
HUTTON, JC ;
PESHAVARIA, M ;
BROCKLEHURST, KW .
BIOCHEMICAL JOURNAL, 1984, 224 (02) :483-490
[6]  
INAGAKI M, 1985, J BIOL CHEM, V260, P2922
[7]  
INAGAKI M, 1984, J BIOL CHEM, V259, P4321
[8]  
KESSEL D, 1985, CANCER RES, V45, P1687
[9]  
KIKKAWA U, 1982, J BIOL CHEM, V257, P13341
[10]   CALCIUM-DEPENDENT PROTEIN-KINASE - WIDESPREAD OCCURRENCE IN VARIOUS TISSUES AND PHYLA OF THE ANIMAL KINGDOM AND COMPARISON OF EFFECTS OF PHOSPHOLIPID, CALMODULIN, AND TRIFLUOPERAZINE [J].
KUO, JF ;
ANDERSSON, RGG ;
WISE, BC ;
MACKERLOVA, L ;
SALOMONSSON, I ;
BRACKETT, NL ;
KATOH, N ;
SHOJI, M ;
WRENN, RW .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (12) :7039-7043