(-)-H-3 DESMETHOXYVERAPAMIL LABELING OF PUTATIVE CALCIUM CHANNELS IN BRAIN - AUTORADIOGRAPHIC DISTRIBUTION AND ALLOSTERIC COUPLING TO 1,4-DIHYDROPYRIDINE AND DILTIAZEM BINDING-SITES

被引:86
作者
FERRY, DR [1 ]
GOLL, A [1 ]
GADOW, C [1 ]
GLOSSMANN, H [1 ]
机构
[1] UNIV GIESSEN,RUDOLF BUCHHEIM INST PHARMAKOL,D-6300 GIESSEN,FED REP GER
关键词
D O I
10.1007/BF00500915
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:183 / 187
页数:5
相关论文
共 19 条
[1]   NOVEL 1,4-DIHYDROPYRIDINE (BAY K-8644) FACILITATES CALCIUM-DEPENDENT [H-3]NORADRENALINE RELEASE FROM PC-12 CELLS [J].
ALBUS, U ;
HABERMANN, E ;
FERRY, DR ;
GLOSSMANN, H .
JOURNAL OF NEUROCHEMISTRY, 1984, 42 (04) :1186-1189
[2]   THE MOLECULAR-BASIS OF NEURONAL EXCITABILITY [J].
CATTERALL, WA .
SCIENCE, 1984, 223 (4637) :653-661
[3]   THE EFFECTS OF LESIONS IN THE RAT HIPPOCAMPUS SUGGEST THE ASSOCIATION OF CALCIUM-CHANNEL BLOCKER BINDING-SITES WITH SPECIFIC NEURONAL POPULATION [J].
CORTES, R ;
SUPAVILAI, P ;
KAROBATH, M ;
PALACIOS, JM .
NEUROSCIENCE LETTERS, 1983, 42 (03) :249-254
[4]   IDENTIFICATION OF PUTATIVE CALCIUM CHANNELS IN SKELETAL-MUSCLE MICROSOMES [J].
FERRY, DR ;
GLOSSMANN, H .
FEBS LETTERS, 1982, 148 (02) :331-337
[5]   EVIDENCE FOR MULTIPLE RECEPTOR-SITES WITHIN THE PUTATIVE CALCIUM-CHANNEL [J].
FERRY, DR ;
GLOSSMANN, H .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 321 (01) :80-83
[6]   [H-3] VERAPAMIL BINDING-SITES IN SKELETAL-MUSCLE TRANSVERSE TUBULE MEMBRANES [J].
GALIZZI, JP ;
FOSSET, M ;
LAZDUNSKI, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 118 (01) :239-245
[7]   CALCIUM CHANNELS - DIRECT IDENTIFICATION WITH RADIOLIGAND BINDING-STUDIES [J].
GLOSSMANN, H ;
FERRY, DR ;
LUBBECKE, F ;
MEWES, R ;
HOFMANN, F .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1982, 3 (11) :431-437
[8]   TEMPERATURE-DEPENDENT REGULATION OF D-CIS-[H-3] DILTIAZEM BINDING TO CA-2+ CHANNELS BY 1,4-DIHYDROPYRIDINE CHANNEL AGONISTS AND ANTAGONISTS [J].
GLOSSMANN, H ;
LINN, T ;
ROMBUSCH, M ;
FERRY, DR .
FEBS LETTERS, 1983, 160 (1-2) :226-232
[9]   TARGET SIZE ANALYSIS AND MOLECULAR-PROPERTIES OF CA-2+ CHANNELS LABELED WITH [H-3] VERAPAMIL [J].
GOLL, A ;
FERRY, DR ;
GLOSSMANN, H .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1984, 141 (01) :177-186
[10]   REVERSIBLE INHIBITION OF POTASSIUM CONTRACTURES BY OPTICAL ISOMERS OF VERAPAMIL AND D 600 ON SLOW MUSCLE-FIBERS OF FROG [J].
KAUMANN, AJ ;
UCHITEL, OD .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1976, 292 (01) :21-27