ENKEPHALIN CONVERTASE - POTENT, SELECTIVE, AND IRREVERSIBLE INHIBITORS

被引:70
作者
FRICKER, LD
PLUMMER, TH
SNYDER, SH
机构
[1] JOHNS HOPKINS UNIV,SCH MED,DEPT PHARMACOL & EXPTL THERAPEUT,BALTIMORE,MD 21205
[2] JOHNS HOPKINS UNIV,SCH MED,DEPT PSYCHIAT & BEHAV SCI,BALTIMORE,MD 21205
[3] NEW YORK STATE DEPT HLTH,CTR LABS & RES,ALBANY,NY 12201
关键词
D O I
10.1016/0006-291X(83)91398-0
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:994 / 1000
页数:7
相关论文
共 8 条
[1]   ENKEPHALIN CONVERTASE - A SPECIFIC ENKEPHALIN SYNTHESIZING CARBOXYPEPTIDASE IN ADRENAL CHROMAFFIN GRANULES, BRAIN, AND PITUITARY-GLAND [J].
FRICKER, LD ;
SUPATTAPONE, S ;
SNYDER, SH .
LIFE SCIENCES, 1982, 31 (16-1) :1841-1844
[2]   ENKEPHALIN CONVERTASE - PURIFICATION AND CHARACTERIZATION OF A SPECIFIC ENKEPHALIN-SYNTHESIZING CARBOXYPEPTIDASE LOCALIZED TO ADRENAL CHROMAFFIN GRANULES [J].
FRICKER, LD ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (12) :3886-3890
[3]  
KIMMEL MT, 1972, J BIOL CHEM, V247, P7864
[4]   BY-PRODUCT ANALOGS FOR BOVINE CARBOXYPEPTIDASE-B [J].
MCKAY, TJ ;
PLUMMER, TH .
BIOCHEMISTRY, 1978, 17 (03) :401-405
[5]   COMPARATIVE STUDIES ON HUMAN CARBOXYPEPTIDASE-B AND CARBOXYPEPTIDASE-N [J].
MCKAY, TJ ;
PHELAN, AW ;
PLUMMER, TH .
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1979, 197 (02) :487-492
[6]   A POTENT MERCAPTO BI-PRODUCT ANALOG INHIBITOR FOR HUMAN CARBOXYPEPTIDASE-N [J].
PLUMMER, TH ;
RYAN, TJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 98 (02) :448-454
[7]  
PLUMMER TH, 1981, FED PROC, V40, P1603
[8]  
SILLEN LG, 1964, SPECIAL PUBLICATION, V17, P364