A NEW CLASS OF INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE

被引:46
作者
HASSALL, CH [1 ]
JOHNSON, WH [1 ]
KENNEDY, AJ [1 ]
ROBERTS, NA [1 ]
机构
[1] ROCHE PROD LTD,WELWYN GARDEN CIT AL7 3AY,HERTS,ENGLAND
关键词
D O I
10.1016/0014-5793(85)80776-6
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:201 / 205
页数:5
相关论文
共 16 条
[1]   ACTIVE SITE OF ELASTASE - PARTIAL MAPPING BY MEANS OF SPECIFIC PEPTIDE SUBSTRATES [J].
ATLAS, D ;
LEVIT, S ;
SCHECHTER, I ;
BERGER, A .
FEBS LETTERS, 1970, 11 (04) :281-+
[2]  
BAGGIOLINI M, 1978, AGENTS ACTIONS, V8, P3, DOI 10.1007/BF01972395
[3]   SYNTHESIS AND ANALYTICAL USE OF A HIGHLY SENSITIVE AND CONVENIENT SUBSTRATE OF ELASTASE [J].
BIETH, J ;
SPIESS, B ;
WERMUTH, CG .
BIOCHEMICAL MEDICINE, 1974, 11 (04) :350-357
[4]   SENSITIVE SUBSTRATES FOR HUMAN-LEUKOCYTE AND PORCINE PANCREATIC ELASTASE - STUDY OF THE MERITS OF VARIOUS CHROMOPHORIC AND FLUOROGENIC LEAVING GROUPS IN ASSAYS FOR SERINE PROTEASES [J].
CASTILLO, MJ ;
NAKAJIMA, K ;
ZIMMERMAN, M ;
POWERS, JC .
ANALYTICAL BIOCHEMISTRY, 1979, 99 (01) :53-64
[5]   SOME NOVEL INHIBITORS OF PORCINE PANCREATIC ELASTASE [J].
HASSALL, CH ;
JOHNSON, WH ;
ROBERTS, NA .
BIOORGANIC CHEMISTRY, 1979, 8 (03) :299-309
[6]  
HASSALL CH, 1980, ENZYME INHIBITORS, P259
[7]  
JANOFF A, 1983, LUNG BIOL HLTH DIS, V19, P173
[8]   NEUTRAL PROTEASES OF HUMAN GRANULOCYTES - ISOLATION AND PARTIAL CHARACTERIZATION OF GRANULOCYTE ELASTASES [J].
OHLSSON, K ;
OLSSON, I .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1974, 42 (02) :519-527
[9]   DRUG ABSORPTION FROM LUNG [J].
SCHANKER, LS .
BIOCHEMICAL PHARMACOLOGY, 1978, 27 (04) :381-385
[10]   ON SIZE OF ACTIVE SITE IN PROTEASES .I. PAPAIN [J].
SCHECHTER, I ;
BERGER, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1967, 27 (02) :157-+