5-HT3 RECEPTORS MEDIATE INHIBITION OF ACETYLCHOLINE-RELEASE IN CORTICAL TISSUE

被引:237
作者
BARNES, JM [1 ]
BARNES, NM [1 ]
COSTALL, B [1 ]
NAYLOR, RJ [1 ]
TYERS, MB [1 ]
机构
[1] GLAXO GRP RES LTD,DEPT NEUROPHARMACOL,WARE SG12 ODP,HERTS,ENGLAND
关键词
D O I
10.1038/338762a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:762 / 763
页数:2
相关论文
共 20 条
[1]  
BARNES JM, IN PRESS BRAIN RES
[2]   [H-3] ZACOPRIDE - LIGAND FOR THE IDENTIFICATION OF 5-HT3 RECOGNITION SITES [J].
BARNES, NM ;
COSTALL, B ;
NAYLOR, RJ .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1988, 40 (08) :548-551
[3]   PHARMACOLOGICAL PROPERTIES OF GR38032F, A NOVEL ANTAGONIST AT 5-HT3 RECEPTORS [J].
BUTLER, A ;
HILL, JM ;
IRELAND, SJ ;
JORDAN, CC ;
TYERS, MB .
BRITISH JOURNAL OF PHARMACOLOGY, 1988, 94 (02) :397-412
[4]   EFFECTS OF THE 5-HT3 RECEPTOR ANTAGONIST, GR38032F, ON RAISED DOPAMINERGIC ACTIVITY IN THE MESOLIMBIC SYSTEM OF THE RAT AND MARMOSET BRAIN [J].
COSTALL, B ;
DOMENEY, AM ;
NAYLOR, RJ ;
TYERS, MB .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 92 (04) :881-894
[5]   ZACOPRIDE - ANXIOLYTIC PROFILE IN RODENT AND PRIMATE MODELS OF ANXIETY [J].
COSTALL, B ;
DOMENEY, AM ;
GERRARD, PA ;
KELLY, ME ;
NAYLOR, RJ .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1988, 40 (04) :302-305
[6]   EFFECT OF QUIPAZINE, A SEROTONIN-LIKE DRUG, ON STRIATAL CHOLINERGIC INTERNEURONES [J].
EUVRARD, C ;
JAVOY, F ;
HERBERT, A ;
GLOWINSKI, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 41 (03) :281-289
[7]   BLOCKADE OF NEURONAL TRYPTAMINE RECEPTORS BY METOCLOPRAMIDE [J].
FOZARD, JR ;
MOBAROKALI, ATM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 49 (01) :109-112
[8]   SEROTONIN INHIBITS ACETYLCHOLINE-RELEASE FROM RAT STRIATUM SLICES - EVIDENCE FOR A PRESYNAPTIC RECEPTOR-MEDIATED EFFECT [J].
GILLET, G ;
AMMOR, S ;
FILLION, G .
JOURNAL OF NEUROCHEMISTRY, 1985, 45 (06) :1687-1691
[9]   EFFECT OF THE 5-HT3 RECEPTOR ANTAGONIST, GR38032F, ON RESPONSES TO INJECTION OF A NEUROKININ AGONIST INTO THE VENTRAL TEGMENTAL AREA OF THE RAT-BRAIN [J].
HAGAN, RM ;
BUTLER, A ;
HILL, JM ;
JORDAN, CC ;
IRELAND, SJ ;
TYERS, MB .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 138 (02) :303-305
[10]  
HOYER DT, 1988, PHARM SCI, V9, P89