L-TRANS-EPOXYSUCCINYL-LEUCYLAMIDO(4-GUANIDINO)BUTANE (E-64) AND ITS ANALOGS AS INHIBITORS OF CYSTEINE PROTEINASES INCLUDING CATHEPSINS B, H AND L

被引：1042

作者：

BARRETT, AJ

KEMBHAVI, AA

BROWN, MA

KIRSCHKE, H

KNIGHT, CG

TAMAI, M

HANADA, K

机构：

[1] MARTIN LUTHER UNIV,INST PHYS CHEM,DDR-402 HALLE,GER DEM REP

[2] TAISHO PHARMACEUT CO LTD,RES LABS,OMIYA,SAITAMA 330,JAPAN

来源：

BIOCHEMICAL JOURNAL | 1982年 / 201卷 / 01期

关键词：

D O I：

10.1042/bj2010189

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：189 / 198

页数：10

共 39 条

[1]

Barrett A. J., 1981, METHODS ENZYMOL, V80, P535

[2] IMPROVED COLOR REAGENT FOR USE IN BARRETTS ASSAY OF CATHEPSIN-B [J].

BARRETT, AJ .

ANALYTICAL BIOCHEMISTRY, 1976, 76 (01) :374-376

[3] FLUORIMETRIC ASSAYS FOR CATHEPSIN-B AND CATHEPSIN-H WITH METHYLCOUMARYLAMIDE SUBSTRATES [J].

BARRETT, AJ .

BIOCHEMICAL JOURNAL, 1980, 187 (03) :909-912

[4] HUMAN CATHEPSIN-B1 - PURIFICATION AND SOME PROPERTIES OF ENZYME [J].

BARRETT, AJ .

BIOCHEMICAL JOURNAL, 1973, 131 (04) :809-+

[5]

BARRETT AJ, 1980, CIBA F S, V75, P1

[6] DETERMINATION OF CONCENTRATION OF HYDROLYTIC ENZYME SOLUTIONS - ALPHA-CHYMOTRYPSIN TRYPSIN PAPAIN ELASTASE SUBTILISIN AND ACETYLCHOLINESTERASE [J].

BENDER, ML ;

BEGUECAN.ML ;

BLAKELEY, RL ;

BRUBACHER, LJ ;

FEDER, J ;

GUNTER, CR ;

KEZDY, FJ ;

KILLHEFFER, JV ;

MARSHALL, TH ;

MILLER, CG ;

ROESKE, RW ;

STOOPS, JK .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1966, 88 (24) :5890-+

[7] MAPPING ACTIVE SITE OF PAPAIN WITH AID OF PEPTIDE SUBSTRATES AND INHIBITORS [J].

BERGER, A ;

SCHECHTER, I .

PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES, 1970, 257 (813) :249-+

[8] REACTIONS OF PAPAIN AND OF LOW-MOLECULAR-WEIGHT THIOLS WITH SOME AROMATIC DISULFIDES - 2,2'-DIPYRIDYL DISULFIDE AS A CONVENIENT ACTIVE-SITE TITRANT FOR PAPAIN EVEN IN PRESENCE OF OTHER THIOLS [J].

BROCKLEHURST, K ;

LITTLE, G .

BIOCHEMICAL JOURNAL, 1973, 133 (01) :67-80

[9] P-NITROPHENYL-P'-GUANIDINOBENZOATE HCL - A NEW ACTIVE SITE TITRANT FOR TRYPSIN [J].

CHASE, T ;

SHAW, E .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1967, 29 (04) :508-&

[10]

ELLIOTT SD, 1970, METHOD ENZYMOL, V19, P252

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