OPIATE BINDING-PROPERTIES OF NATURALLY-OCCURRING N-TERMINAL AND C-TERMINAL MODIFIED BETA-ENDORPHINS

被引:150
作者
AKIL, H
YOUNG, E
WATSON, SJ
COY, DH
机构
[1] VET ADM MED CTR, NEW ORLEANS, LA 70146 USA
[2] TULANE UNIV, SCH MED, NEW ORLEANS, LA 70118 USA
关键词
D O I
10.1016/S0196-9781(81)80121-0
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:289 / 292
页数:4
相关论文
共 24 条
[1]   BINDING OF BETA-ENDORPHIN-H-3 TO RAT-BRAIN MEMBRANES - CHARACTERIZATION OF OPIATE PROPERTIES AND INTERACTION WITH ACTH [J].
AKIL, H ;
HEWLETT, WA ;
BARCHAS, JD ;
LI, CH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 64 (01) :1-8
[2]   APPEARANCE OF BETA-ENDORPHIN-LIKE IMMUNOREACTIVITY IN HUMAN VENTRICULAR CEREBROSPINAL-FLUID UPON ANALGESIC ELECTRICAL-STIMULATION [J].
AKIL, H ;
RICHARDSON, DE ;
BARCHAS, JD ;
LI, CH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1978, 75 (10) :5170-5172
[3]   NEURONS CONTAINING BETA-ENDORPHIN IN RAT-BRAIN EXIST SEPARATELY FROM THOSE CONTAINING ENKEPHALIN - IMMUNOCYTOCHEMICAL STUDIES [J].
BLOOM, F ;
BATTENBERG, E ;
ROSSIER, J ;
LING, N ;
GUILLEMIN, R .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1978, 75 (03) :1591-1595
[4]   C FRAGMENT OF LIPOTROPIN HAS A HIGH AFFINITY FOR BRAIN OPIATE RECEPTORS [J].
BRADBURY, AF ;
SMYTH, DG ;
SNELL, CR ;
BIRDSALL, NJM ;
HULME, EC .
NATURE, 1976, 260 (5554) :793-795
[5]  
CHANG KJ, 1979, MOL PHARMACOL, V16, P91
[6]   ISOLATION OF PEPTIDES WITH OPIATE ACTIVITY FROM SHEEP AND HUMAN PITUITARIES - RELATIONSHIP TO BETA-LIPOTROPIN [J].
CHRETIEN, M ;
BENJANNET, S ;
DRAGON, N ;
SEIDAH, NG ;
LIS, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1976, 72 (02) :472-478
[7]   OPIOID ACTIVITY OF A PEPTIDE, BETA-LIPOTROPIN-(61-91), DERIVED FROM BETA-LIPOTROPIN [J].
COX, BM ;
GOLDSTEIN, A ;
LI, CH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1976, 73 (06) :1821-1823
[8]  
COY DH, 1977, 5TH P ANN PEPT S, P107
[9]   INFLUENCE OF N-TERMINAL ACETYLATION AND C-TERMINAL PROTEOLYSIS ON THE ANALGESIC ACTIVITY OF BETA-ENDORPHIN [J].
DEAKIN, JFW ;
DOSTROVSKY, JO ;
SMYTH, DG .
BIOCHEMICAL JOURNAL, 1980, 189 (03) :501-506
[10]  
EIPPER BA, J BIOCH