The structure of thrombin, a chameleon-like proteinase

被引:32
作者
Bode, W [1 ]
机构
[1] Max Planck Inst Biochem, Proteinase Res Grp, D-82152 Martinsried, Germany
关键词
antithrombotics; coagulation; crystal structures; inhibition; thrombin; zymogen activation;
D O I
10.1111/j.1538-7836.2005.01356.x
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:2379 / 2388
页数:10
相关论文
共 101 条
[1]   The crystal structure of activated protein C-inactivated bovine factor Va: Implications for cofactor function [J].
Adams, TE ;
Hockin, MF ;
Mann, KG ;
Everse, SJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2004, 101 (24) :8918-8923
[2]   STRUCTURE OF THE NONCOVALENT COMPLEX OF PROTHROMBIN KRINGLE-2 WITH PPACK-THROMBIN [J].
ARNI, RK ;
PADMANABHAN, K ;
PADMANABHAN, KP ;
WU, TP ;
TULINSKY, A .
CHEMISTRY AND PHYSICS OF LIPIDS, 1994, 67-8 :59-66
[3]   PROTEINASE-INHIBITORS FROM THE EUROPEAN MEDICINAL LEECH HIRUDO-MEDICINALIS STRUCTURAL, FUNCTIONAL AND BIOMEDICAL ASPECTS [J].
ASCENZI, P ;
AMICONI, G ;
BODE, W ;
BOLOGNESI, M ;
COLETTA, M ;
MENEGATTI, E .
MOLECULAR ASPECTS OF MEDICINE, 1995, 16 (03) :215-313
[4]   BINDING OF THE BOVINE BASIC PANCREATIC TRYPSIN-INHIBITOR (KUNITZ) TO HUMAN ALPHA-THROMBIN, BETA-THROMBIN AND GAMMA-THROMBIN - A KINETIC AND THERMODYNAMIC STUDY [J].
ASCENZI, P ;
COLETTA, M ;
AMICONI, G ;
DECRISTOFARO, R ;
BOLOGNESI, M ;
GUARNERI, M ;
MENEGATTI, E .
BIOCHIMICA ET BIOPHYSICA ACTA, 1988, 956 (02) :156-161
[5]   Crystal structures of native and thrombin-complexed heparin cofactor II reveal a multistep allosteric mechanism [J].
Baglin, TP ;
Carrell, RW ;
Church, FC ;
Esmon, CT ;
Huntington, JA .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2002, 99 (17) :11079-11084
[6]  
BAJUSZ S, 1978, INT J PEPT PROT RES, V12, P217
[7]  
BANNER DW, 1991, J BIOL CHEM, V266, P20085
[8]   The crystal structure of the complex of blood coagulation factor VIIa with soluble tissue factor [J].
Banner, DW ;
DArcy, A ;
Chene, C ;
Winkler, FK ;
Guha, A ;
Konigsberg, WH ;
Nemerson, Y ;
Kirchhofer, D .
NATURE, 1996, 380 (6569) :41-46
[9]   Structure of the fifth EGF-like domain of thrombomodulin: An EGF-like domain with a novel disulfide-bonding pattern [J].
Benitez, BAS ;
Hunter, MJ ;
Meininger, DP ;
Komives, EA .
JOURNAL OF MOLECULAR BIOLOGY, 1997, 273 (04) :913-926
[10]   The Protein Data Bank [J].
Berman, HM ;
Westbrook, J ;
Feng, Z ;
Gilliland, G ;
Bhat, TN ;
Weissig, H ;
Shindyalov, IN ;
Bourne, PE .
NUCLEIC ACIDS RESEARCH, 2000, 28 (01) :235-242