STRUCTURE-ACTIVITY-RELATIONSHIPS OF ENKEPHALIN ANALOGS AT OPIATE AND ENKEPHALIN RECEPTORS - CORRELATION WITH ANALGESIA

被引：61

作者：

AUDIGIER, Y

MAZARGUIL, H

GOUT, R

CROS, J

机构：

来源：

EUROPEAN JOURNAL OF PHARMACOLOGY | 1980年 / 63卷 / 01期

关键词：

D O I：

10.1016/0014-2999(80)90114-4

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：35 / 46

页数：12

共 33 条

[1] BINDING OF LEUKENCEPHALIN-H-3 IN RAT STRIATUM - PARTIAL INHIBITION BY MORPHINE OR NALOXONE [J].

AUDIGIER, Y ;

MALFROYCAMINE, B ;

SCHWARTZ, JC .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 41 (02) :247-248

[2] SUPERACTIVE ANTINOCICEPTIVE PENTAPEPTIDE, (D-MET2,PRO5), ENKEPHALINAMIDE [J].

BAJUSZ, S ;

RONAI, AZ ;

SZEKELY, JI ;

GRAF, L ;

DUNAIKOVACS, Z ;

BERZETEI, I .

FEBS LETTERS, 1977, 76 (01) :91-92

[3]

BAJUSZ S, 1978, BIOCHEM BIOPH RES CO, V84, P1045, DOI 10.1016/0006-291X(78)91689-3

[4] ENHANCED ANALGESIC ACTIVITY OF D-ALA2 ENKEPHALINAMIDES FOLLOWING D-ISOMER SUBSTITUTIONS AT POSITION 5 [J].

BELLUZZI, JD ;

STEIN, L ;

DVONCH, W ;

DHEER, S ;

GLUCKMAN, MI ;

MCGREGOR, WH .

LIFE SCIENCES, 1978, 23 (02) :99-104

[5] EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE [J].

BUSCHER, HH ;

HILL, RC ;

ROMER, D ;

CARDINAUX, F ;

CLOSSE, A ;

HAUSER, D ;

PLESS, J .

NATURE, 1976, 261 (5559) :423-425

[6]

CHANG KJ, 1979, J BIOL CHEM, V254, P2610

[7] OPIATE RECEPTOR-BINDING AFFECTED DIFFERENTIALLY BY OPIATES AND OPIOID PEPTIDES [J].

CHILDERS, SR ;

CREESE, I ;

SNOWMAN, AM ;

SNYDER, SH .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (01) :11-18

[8]

D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74

[9]

Della Bella D, 1978, Adv Biochem Psychopharmacol, V18, P271

[10]

GILBERT PE, 1976, J PHARMACOL EXP THER, V198, P66

← 1 2 3 4 →