GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS

被引：140

作者：

BRAESTRUP, C ^{[1
]}

NIELSEN, M ^{[1
]}

机构：

[1] AS FERROSAN,DIV RES,DK-2860 SOEBORG,DENMARK

来源：

NATURE | 1981年 / 294卷 / 5840期

关键词：

D O I：

10.1038/294472a0

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：472 / 474

页数：3

共 14 条

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[2] [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS [J].

BRAESTRUP, C ;

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[3] PARTIAL AGONISTS FOR BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].

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NATURE, 1979, 280 (5720) :331-333

[4] URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS [J].

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[5] ETHYL BETA-CARBOLINE CARBOXYLATE LOWERS SEIZURE THRESHOLD AND ANTAGONIZES FLURAZEPAM-INDUCED SEDATION IN RATS [J].

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[6] GAMMA-AMINOBUTYRIC ACID REGULATION OF THE BENZODIAZEPINE RECEPTOR - BIOCHEMICAL-EVIDENCE FOR PHARMACOLOGICALLY DIFFERENT EFFECTS OF BENZODIAZEPINES AND PROPYL BETA-CARBOLINE-3-CARBOXYLATE [J].

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EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (04) :593-595

[7] SYNTHETIC NON-BENZODIAZEPINE LIGAND FOR BENZODIAZEPINE RECEPTORS - PROBE FOR INVESTIGATING NEURONAL SUBSTRATES OF ANXIETY [J].

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BEER, B .

PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1979, 11 (01) :99-106

[8] PROPERTIES OF DIAZEPAM-H-3 BINDING TO BENZODIAZEPINE RECEPTORS IN RAT CEREBRAL-CORTEX [J].

MOHLER, H ;

OKADA, T .

LIFE SCIENCES, 1977, 20 (12) :2101-2110

[9] [PROPYL-H-3 BETA-CARBOLINE-3-CARBOXYLATE BINDS SPECIFICALLY TO BRAIN BENZODIAZEPINE RECEPTORS [J].

NIELSEN, M ;

SCHOU, H ;

BRAESTRUP, C .

JOURNAL OF NEUROCHEMISTRY, 1981, 36 (01) :276-285

[10] THE PROCONVULSANT AND DIAZEPAM-REVERSING EFFECTS OF ETHYL-BETA-CARBOLINE-3-CARBOXYLATE [J].

OAKLEY, NR ;

JONES, BJ .

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