COMPETITIVE INHIBITION OF SPECIFIC STEROID-PROTEIN BINDING - PRACTICAL USE OF RELATIVE COMPETITION RATIOS FOR THE DERIVATION OF EQUILIBRIUM INHIBITION CONSTANTS

被引:15
作者
BLONDEAU, JP
ROCHER, P
ROBEL, P
机构
关键词
D O I
10.1016/0039-128X(78)90068-5
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:563 / 575
页数:13
相关论文
共 14 条
[1]   COMPARISON OF 7 METHODS FOR FITTING MICHAELIS-MENTEN EQUATION [J].
ATKINS, GL ;
NIMMO, IA .
BIOCHEMICAL JOURNAL, 1975, 149 (03) :775-777
[2]  
BAULIEU EE, 1969, PROGR BIOCHEM PHARMA, V5, P46
[3]   COMPETITIVE INHIBITION - NEW AND GENERAL LINEAR RELATIONS [J].
BESTBELPOMME, M ;
DESSEN, P .
BIOCHIMIE, 1973, 55 (01) :11-16
[4]   DETERMINATION OF PROTEIN-LIGAND BINDING CONSTANTS AT EQUILIBRIUM IN BIOLOGICAL SAMPLES [J].
BLONDEAU, JP ;
ROBEL, P .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1975, 55 (02) :375-384
[5]   THE EFFECT OF PH ON THE AFFINITIES OF ENZYMES FOR SUBSTRATES AND INHIBITORS [J].
DIXON, M .
BIOCHEMICAL JOURNAL, 1953, 55 (01) :161-170
[6]  
Eadie GS, 1942, J BIOL CHEM, V146, P85
[7]  
EDSALL JT, 1958, BIOPHYS CHEM, V1, P591
[8]   DETERMINATION, AT EQUILIBRIUM, OF ASSOCIATION CONSTANTS OF LABELED OR UNLABELLED LIGANDS BY A NON-GRAPHICAL METHOD [J].
GOERTZ, G ;
LONGCHAMPT, J ;
CREPY, O ;
JUDAS, O ;
JAYLE, MF .
BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 451 (01) :287-304
[9]  
KORENMAN SG, 1970, ACTA ENDOCRINOL-COP, P291
[10]   The determination of enzyme dissociation constants [J].
Lineweaver, H ;
Burk, D .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1934, 56 :658-666