[BE-2254-I-125, A NEW HIGH-AFFINITY RADIOLIGAND FOR ALPHA-1-ADRENOCEPTORS

被引:177
作者
ENGEL, G
HOYER, D
机构
关键词
D O I
10.1016/0014-2999(81)90095-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
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页码:221 / 224
页数:4
相关论文
共 12 条
[1]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[2]  
Engel G, 1980, Triangle, V19, P69
[3]   THE USE OF LIGAND-BINDING FOR THE CHARACTERIZATION OF ALPHA-ADRENOCEPTORS [J].
GLOSSMANN, H ;
HORNUNG, R ;
PRESEK, P .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1980, 2 :S303-S324
[4]   PREFERENTIAL BLOCKADE OF POSTSYNAPTIC ALPHA-ADRENOCEPTORS BY BE-2254 [J].
GOTHERT, M ;
NOLTE, J ;
WEINHEIMER, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (01) :35-42
[5]   BINDING CHARACTERISTICS OF PRAZOSIN-H-3 TO RAT-BRAIN ALPHA-ADRENERGIC RECEPTORS [J].
GREENGRASS, P ;
BREMNER, R .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (03) :323-326
[6]   FUNCTIONAL-CHARACTERIZATION OF CENTRAL ALPHA-ADRENOCEPTORS BY YOHIMBINE DIASTEREOMERS [J].
HEDLER, L ;
STAMM, G ;
WEITZELL, R ;
STARKE, K .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (01) :43-52
[7]  
HEINZ N, 1980, ARZNEIMITTEL-FORSCH, V30-2, P2135
[8]   ALPHA-ADRENOCEPTORS IN RAT-BRAIN - DIRECT IDENTIFICATION WITH PRAZOSIN [J].
HORNUNG, R ;
PRESEK, P ;
GLOSSMANN, H .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 308 (03) :223-230
[9]   DISTINCT ALPHA-NORADRENERGIC RECEPTORS DIFFERENTIATED BY BINDING AND PHYSIOLOGICAL RELATIONSHIPS [J].
PRICHARD, DCU ;
SNYDER, SH .
LIFE SCIENCES, 1979, 24 (01) :79-88
[10]   THE ATTRACTIONS OF PROTEINS FOR SMALL MOLECULES AND IONS [J].
SCATCHARD, G .
ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1949, 51 (04) :660-672