IONIC REQUIREMENTS FOR THE SPECIFIC BINDING OF [H-3]GBR 12783 TO A SITE ASSOCIATED WITH THE DOPAMINE UPTAKE CARRIER

被引:37
作者
BONNET, JJ
BENMANSOUR, S
VAUGEOIS, JM
COSTENTIN, J
机构
关键词
D O I
10.1111/j.1471-4159.1988.tb02979.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:759 / 765
页数:7
相关论文
共 18 条
[1]   SODIUM INDEPENDENCE OF THE BINDING OF [H-3] GBR 12783 AND OTHER DOPAMINE UPTAKE INHIBITORS TO THE DOPAMINE UPTAKE COMPLEX [J].
BENMANSOUR, S ;
BONNET, JJ ;
PROTAIS, P ;
COSTENTIN, J .
NEUROSCIENCE LETTERS, 1987, 77 (01) :97-102
[2]   MEMBRANE-POTENTIALS IN PINCHED-OFF PRESYNAPTIC NERVE-TERMINALS MONITORED WITH A FLUORESCENT-PROBE - EVIDENCE THAT SYNAPTOSOMES HAVE POTASSIUM DIFFUSION POTENTIALS [J].
BLAUSTEIN, MP ;
GOLDRING, JM .
JOURNAL OF PHYSIOLOGY-LONDON, 1975, 247 (03) :589-615
[3]   HIGH-AFFINITY [H-3] GBR 12783 BINDING TO A SPECIFIC SITE ASSOCIATED WITH THE NEURONAL DOPAMINE UPTAKE COMPLEX IN THE CENTRAL-NERVOUS-SYSTEM [J].
BONNET, JJ ;
PROTAIS, P ;
CHAGRAOUI, A ;
COSTENTIN, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) :211-222
[4]   GBR-12783, A POTENT AND SELECTIVE INHIBITOR OF DOPAMINE UPTAKE - BIOCHEMICAL-STUDIES INVIVO AND EXVIVO [J].
BONNET, JJ ;
COSTENTIN, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 121 (02) :199-209
[5]   BINDING CHARACTERISTICS OF THE DOPAMINE UPTAKE INHIBITOR [H-3] NOMIFENSINE TO STRIATAL MEMBRANES [J].
DUBOCOVICH, ML ;
ZAHNISER, NR .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (08) :1137-1144
[6]  
FISCHER JF, 1979, J PHARMACOL EXP THER, V208, P203
[7]  
HOLZ RW, 1974, MOL PHARMACOL, V10, P746
[8]   CHARACTERIZATION OF SODIUM-DEPENDENT [H-3] GBR-12935 BINDING IN BRAIN - A RADIOLIGAND FOR SELECTIVE LABELING OF THE DOPAMINE TRANSPORT COMPLEX [J].
JANOWSKY, A ;
BERGER, P ;
VOCCI, F ;
LABARCA, R ;
SKOLNICK, P ;
PAUL, SM .
JOURNAL OF NEUROCHEMISTRY, 1986, 46 (04) :1272-1276
[9]  
JAVITCH JA, 1984, MOL PHARMACOL, V26, P35
[10]   SODIUM-SENSITIVE COCAINE BINDING TO RAT STRIATAL MEMBRANE - POSSIBLE RELATIONSHIP TO DOPAMINE UPTAKE SITES [J].
KENNEDY, LT ;
HANBAUER, I .
JOURNAL OF NEUROCHEMISTRY, 1983, 41 (01) :172-178