TYPE-I AND TYPE-II GABAA-BENZODIAZEPINE RECEPTORS PRODUCED IN TRANSFECTED CELLS

被引:741
作者
PRITCHETT, DB
LUDDENS, H
SEEBURG, PH
机构
关键词
D O I
10.1126/science.2551039
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:1389 / 1392
页数:4
相关论文
共 41 条
[1]   SELECTIVE AFFINITY OF THE BENZODIAZEPINES QUAZEPAM AND 2-OXO-QUAZEPAM FOR BZ1 BINDING-SITE AND DEMONSTRATION OF H-3-2-OXO-QUAZEPAM AS A BZ1 SELECTIVE RADIOLIGAND [J].
BILLARD, W ;
CROSBY, G ;
IORIO, L ;
CHIPKIN, R ;
BARNETT, A .
LIFE SCIENCES, 1988, 42 (02) :179-187
[2]  
CASALOTTI SO, 1986, J BIOL CHEM, V261, P5013
[3]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[4]   PREFERENTIAL AFFINITY OF H-3-2-OXO-QUAZEPAM FOR TYPE-I BENZODIAZEPINE RECOGNITION SITES IN THE HUMAN-BRAIN [J].
CORDA, MG ;
GIORGI, O ;
LONGONI, B ;
ONGINI, E ;
MONTALDO, S ;
BIGGIO, G .
LIFE SCIENCES, 1988, 42 (02) :189-197
[5]   DIFFERENTIAL DEGRADATION OF DIFFERENT BENZODIAZEPINE BINDING-PROTEINS BY INCUBATION OF MEMBRANES FROM CEREBELLUM OR HIPPOCAMPUS WITH TRYPSIN [J].
EICHINGER, A ;
SIEGHART, W .
JOURNAL OF NEUROCHEMISTRY, 1985, 45 (01) :219-226
[6]   PHOTOAFFINITY-LABELING OF DIFFERENT BENZODIAZEPINE RECEPTORS AT PHYSIOLOGICAL TEMPERATURE [J].
EICHINGER, A ;
SIEGHART, W .
JOURNAL OF NEUROCHEMISTRY, 1984, 43 (06) :1745-1748
[7]   VARIOUS PROTEINS FROM RAT-BRAIN, SPECIFICALLY AND IRREVERSIBLY LABELED BY [H-3]FLUNITRAZEPAM, ARE DISTINCT ALPHA-SUBUNITS OF THE GABA BENZODIAZEPINE RECEPTOR COMPLEX [J].
FUCHS, K ;
MOHLER, H ;
SIEGHART, W .
NEUROSCIENCE LETTERS, 1988, 90 (03) :314-319
[8]   REGIONAL HETEROGENEITY OF BENZODIAZEPINE RECEPTORS AT 37-DEGREES-C - AN INVITRO STUDY IN VARIOUS REGIONS OF THE RAT-BRAIN [J].
GEE, KW ;
YAMAMURA, HI .
LIFE SCIENCES, 1982, 31 (18) :1939-1945
[9]   THE INFLUENCE OF TEMPERATURE AND GAMMA-AMINOBUTYRIC ACID ON BENZODIAZEPINE RECEPTOR SUBTYPES IN THE HIPPOCAMPUS OF THE RAT [J].
GEE, KW ;
EHLERT, FJ ;
YAMAMURA, HI .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 106 (04) :1134-1140