STEREOSELECTIVE METABOLISM OF THE 5-LIPOXYGENASE INHIBITOR A-78773

被引:5
作者
CARTER, GW
BELL, RL
MARSH, K
LANNI, C
AWNI, WM
BOUSKA, J
STEWART, AO
HANSEN, R
DUBE, L
BROOKS, DW
机构
来源
CELLULAR GENERATION, TRANSPORT, AND EFFECTS OF EICOSANOIDS: BIOLOGICAL ROLES AND PHARMACOLOGICAL INTERVENTION | 1994年 / 744卷
关键词
D O I
10.1111/j.1749-6632.1994.tb52744.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:262 / 273
页数:12
相关论文
共 32 条
[1]   THE EFFECT OF AN INHALED LEUKOTRIENE ANTAGONIST, L-648,051, ON EARLY AND LATE ASTHMATIC REACTIONS AND SUBSEQUENT INCREASE IN AIRWAY RESPONSIVENESS IN MAN [J].
BEL, EH ;
TIMMERS, MC ;
DIJKMAN, JH ;
STAHL, EG ;
STERK, PJ .
JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 1990, 85 (06) :1067-1075
[2]   THE PROPERTIES OF A-69412 - A SMALL HYDROPHILIC 5-LIPOXYGENASE INHIBITOR [J].
BELL, RL ;
BOUSKA, J ;
YOUNG, PR ;
LANNI, C ;
MACHINIST, J ;
MALO, PE ;
SUMMERS, JB ;
BROOKS, DW ;
CARTER, GW .
AGENTS AND ACTIONS, 1993, 38 (3-4) :178-187
[3]  
BELL RL, 1993, J LIPID MEDIATOR, V6, P259
[4]  
Britton J, 1987, Adv Prostaglandin Thromboxane Leukot Res, V17B, P1003
[5]  
CARTER GW, 1991, J PHARMACOL EXP THER, V256, P929
[6]   THE POTENT AND SELECTIVE SULFIDOPEPTIDE LEUKOTRIENE ANTAGONIST, SK-AND-F-104353, INHIBITS ASPIRIN-INDUCED ASTHMA [J].
CHRISTIE, PE ;
SMITH, CM ;
LEE, TH .
AMERICAN REVIEW OF RESPIRATORY DISEASE, 1991, 144 (04) :957-958
[7]   A SPECIFIC LTD4 LTE4-RECEPTOR ANTAGONIST IMPROVES PULMONARY-FUNCTION IN PATIENTS WITH MILD, CHRONIC ASTHMA [J].
CLOUD, ML ;
ENAS, GC ;
KEMP, J ;
PLATTSMILLS, T ;
ALTMAN, LC ;
TOWNLEY, R ;
TINKELMAN, D ;
KING, T ;
MIDDLETON, E ;
SHEFFER, AL ;
MCFADDEN, ER ;
FARLOW, DS .
AMERICAN REVIEW OF RESPIRATORY DISEASE, 1989, 140 (05) :1336-1339
[8]  
DAHLEN B, 1993, EUR RESPIR J, V6, P1018
[9]  
DAHLEN SE, 1991, ADV PROSTAG THROMB L, V21, P461
[10]   EFFECT OF THE ORAL LEUKOTRIENE ANTAGONIST, ICI 204,219, ON ANTIGEN-INDUCED BRONCHOCONSTRICTION IN SUBJECTS WITH ASTHMA [J].
FINDLAY, SR ;
BARDEN, JM ;
EASLEY, CB ;
GLASS, M .
JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 1992, 89 (05) :1040-1045