BETA-RECEPTOR OCCUPANCY - ASSESSMENT IN THE INTACT ANIMAL

被引:16
作者
HOMCY, CJ
STRAUSS, HW
KOPIWODA, S
机构
[1] MASSACHUSETTS GEN HOSP,DEPT RADIOL,DIV NUCL MED,BOSTON,MA 02114
[2] HARVARD UNIV,MASSACHUSETTS GEN HOSP,SCH MED,BOSTON,MA 02114
关键词
D O I
10.1172/JCI109764
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1111 / 1118
页数:8
相关论文
共 25 条
[1]   ISOPRENALINE-INDUCED AND EXERCISE-INDUCED TACHYCARDIA IN ASSESSMENT OF BETA/ADRENOCEPTOR BLOCKING-DRUGS - COMPARISON BETWEEN TOLAMOLOL, PRACTOLOL AND PROPRANOLOL [J].
ADAM, KR ;
PULLMAN, LG ;
SCHOLFIELD, PC .
BRITISH JOURNAL OF PHARMACOLOGY, 1973, 49 (03) :560-563
[2]  
ANSARI AN, 1974, CARDIOVASCULAR NUCLE, P234
[3]   BETA-ADRENERGIC-RECEPTOR - STEREOSPECIFIC INTERACTION OF IODINATED BETA-BLOCKING AGENT WITH HIGH AFFINITY SITE [J].
AURBACH, GD ;
FEDAK, SA ;
WOODARD, CJ ;
PALMER, JS .
SCIENCE, 1974, 186 (4170) :1223-1224
[4]   NORADRENALINE - FATE AND CONTROL OF ITS BIOSYNTHESIS [J].
AXELROD, J .
SCIENCE, 1971, 173 (3997) :598-+
[5]  
BROWN EA, 1976, J BIOL CHEM, V254, P1239
[6]  
BYLUND DB, 1977, J PHARMACOL EXP THER, V201, P644
[7]  
Cuatrecasas P, 1976, Adv Protein Chem, V30, P251, DOI 10.1016/S0065-3233(08)60481-7
[8]   NORADRENALINE BINDING AND SEARCH FOR CATECHOLAMINE RECEPTORS [J].
CUATRECASAS, P ;
TELL, GPE ;
SICA, V ;
PARIKH, I ;
CHANG, KJ .
NATURE, 1974, 247 (5436) :92-97
[9]   SIMULTANEOUS RADIOENZYMATIC DETERMINATION OF PLASMA AND TISSUE ADRENALINE, NORADRENALINE AND DOPAMINE WITHIN FEMTOMOLE RANGE [J].
DAPRADA, M ;
ZURCHER, G .
LIFE SCIENCES, 1976, 19 (08) :1161-1174
[10]   ELEVATED BETA-ADRENERGIC-RECEPTOR NUMBER AFTER CHRONIC PROPRANOLOL TREATMENT [J].
GLAUBIGER, G ;
LEFKOWITZ, RJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 78 (02) :720-725