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BENZODIAZEPINE GASTRIN AND BRAIN CHOLECYSTOKININ RECEPTOR LIGANDS - L-365,260
被引:351
作者
:
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
BOCK, MG
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
DIPARDO, RM
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
EVANS, BE
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
RITTLE, KE
WHITTER, WL
论文数:
0
引用数:
0
h-index:
0
WHITTER, WL
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
VEBER, DF
ANDERSON, PS
论文数:
0
引用数:
0
h-index:
0
ANDERSON, PS
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
FREIDINGER, RM
机构
:
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1989年
/ 32卷
/ 01期
关键词
:
D O I
:
10.1021/jm00121a004
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:13 / 16
页数:4
相关论文
共 18 条
[1]
CHOLECYSTOKININ IN THE CENTRAL NERVOUS-SYSTEM - A MINIREVIEW
[J].
BEINFELD, MC
论文数:
0
引用数:
0
h-index:
0
BEINFELD, MC
.
NEUROPEPTIDES,
1983,
3
(06)
:411
-427
[2]
AN EXPEDIENT SYNTHESIS OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONE
[J].
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
BOCK, MG
;
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
DIPARDO, RM
;
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
EVANS, BE
;
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
RITTLE, KE
;
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
VEBER, DF
;
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
FREIDINGER, RM
.
TETRAHEDRON LETTERS,
1987,
28
(09)
:939
-942
[3]
SYNTHESIS AND RESOLUTION OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONES
[J].
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
BOCK, MG
;
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
DIPARDO, RM
;
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
EVANS, BE
;
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
RITTLE, KE
;
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
VEBER, DF
;
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
FREIDINGER, RM
;
HIRSHFIELD, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
HIRSHFIELD, J
;
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
SPRINGER, JP
.
JOURNAL OF ORGANIC CHEMISTRY,
1987,
52
(15)
:3232
-3239
[4]
CHARACTERIZATION OF [H-3] PENTAGASTRIN BINDING IN GUINEA-PIG GASTRIC GLANDS - AN ALTERNATIVE CONVENIENT LIGAND FOR RECEPTOR-BINDING ASSAY
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
LOTTI, VJ
;
KEEGAN, ME
论文数:
0
引用数:
0
h-index:
0
KEEGAN, ME
;
KUNKEL, KA
论文数:
0
引用数:
0
h-index:
0
KUNKEL, KA
.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1986,
134
(02)
:895
-899
[5]
TIFLUADOM, A KAPPA-OPIATE AGONIST, ACTS AS A PERIPHERAL CHOLECYSTOKININ RECEPTOR ANTAGONIST
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
LOTTI, VJ
;
CHEN, TB
论文数:
0
引用数:
0
h-index:
0
CHEN, TB
;
KEEGAN, ME
论文数:
0
引用数:
0
h-index:
0
KEEGAN, ME
.
NEUROSCIENCE LETTERS,
1986,
72
(02)
:211
-214
[6]
BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF AN EXTREMELY POTENT AND SELECTIVE NONPEPTIDE CHOLECYSTOKININ ANTAGONIST
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
LOTTI, VJ
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1986,
83
(13)
:4923
-4926
[7]
A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
LOTTI, VJ
;
MONAGHAN, RL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
MONAGHAN, RL
;
BIRNBAUM, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
BIRNBAUM, J
;
STAPLEY, EO
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
STAPLEY, EO
;
GOETZ, MA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
GOETZ, MA
;
ALBERSSCHONBERG, G
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
ALBERSSCHONBERG, G
;
PATCHETT, AA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
PATCHETT, AA
;
LIESCH, JM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
LIESCH, JM
;
HENSENS, OD
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
HENSENS, OD
;
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
SPRINGER, JP
.
SCIENCE,
1985,
230
(4722)
:177
-179
[8]
CYCLIC CHOLECYSTOKININ ANALOGS WITH HIGH SELECTIVITY FOR CENTRAL RECEPTORS
[J].
CHARPENTIER, B
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
CHARPENTIER, B
;
PELAPRAT, D
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
PELAPRAT, D
;
DURIEUX, C
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
DURIEUX, C
;
DOR, A
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
DOR, A
;
REIBAUD, M
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
REIBAUD, M
;
BLANCHARD, JC
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
BLANCHARD, JC
;
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, DEPT CHIM ORGAN,CNRS,UNITE 498,INSERM,U266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
ROQUES, BP
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1988,
85
(06)
:1968
-1972
[9]
DESIGN OF POTENT, ORALLY EFFECTIVE, NONPEPTIDAL ANTAGONISTS OF THE PEPTIDE-HORMONE CHOLECYSTOKININ
[J].
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
EVANS, BE
;
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
BOCK, MG
;
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
RITTLE, KE
;
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
DIPARDO, RM
;
WHITTER, WL
论文数:
0
引用数:
0
h-index:
0
WHITTER, WL
;
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
VEBER, DF
;
ANDERSON, PS
论文数:
0
引用数:
0
h-index:
0
ANDERSON, PS
;
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
FREIDINGER, RM
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1986,
83
(13)
:4918
-4922
[10]
EVANS BE, 1988, J MED CHEM, V32, P2235
←
1
2
→
共 18 条
[1]
CHOLECYSTOKININ IN THE CENTRAL NERVOUS-SYSTEM - A MINIREVIEW
[J].
BEINFELD, MC
论文数:
0
引用数:
0
h-index:
0
BEINFELD, MC
.
NEUROPEPTIDES,
1983,
3
(06)
:411
-427
[2]
AN EXPEDIENT SYNTHESIS OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONE
[J].
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
BOCK, MG
;
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
DIPARDO, RM
;
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
EVANS, BE
;
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
RITTLE, KE
;
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
VEBER, DF
;
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
FREIDINGER, RM
.
TETRAHEDRON LETTERS,
1987,
28
(09)
:939
-942
[3]
SYNTHESIS AND RESOLUTION OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONES
[J].
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
BOCK, MG
;
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
DIPARDO, RM
;
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
EVANS, BE
;
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
RITTLE, KE
;
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
VEBER, DF
;
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
FREIDINGER, RM
;
HIRSHFIELD, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
HIRSHFIELD, J
;
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
SPRINGER, JP
.
JOURNAL OF ORGANIC CHEMISTRY,
1987,
52
(15)
:3232
-3239
[4]
CHARACTERIZATION OF [H-3] PENTAGASTRIN BINDING IN GUINEA-PIG GASTRIC GLANDS - AN ALTERNATIVE CONVENIENT LIGAND FOR RECEPTOR-BINDING ASSAY
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
LOTTI, VJ
;
KEEGAN, ME
论文数:
0
引用数:
0
h-index:
0
KEEGAN, ME
;
KUNKEL, KA
论文数:
0
引用数:
0
h-index:
0
KUNKEL, KA
.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1986,
134
(02)
:895
-899
[5]
TIFLUADOM, A KAPPA-OPIATE AGONIST, ACTS AS A PERIPHERAL CHOLECYSTOKININ RECEPTOR ANTAGONIST
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
LOTTI, VJ
;
CHEN, TB
论文数:
0
引用数:
0
h-index:
0
CHEN, TB
;
KEEGAN, ME
论文数:
0
引用数:
0
h-index:
0
KEEGAN, ME
.
NEUROSCIENCE LETTERS,
1986,
72
(02)
:211
-214
[6]
BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF AN EXTREMELY POTENT AND SELECTIVE NONPEPTIDE CHOLECYSTOKININ ANTAGONIST
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
LOTTI, VJ
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1986,
83
(13)
:4923
-4926
[7]
A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS
[J].
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
CHANG, RSL
;
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
LOTTI, VJ
;
MONAGHAN, RL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
MONAGHAN, RL
;
BIRNBAUM, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
BIRNBAUM, J
;
STAPLEY, EO
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
STAPLEY, EO
;
GOETZ, MA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
GOETZ, MA
;
ALBERSSCHONBERG, G
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
ALBERSSCHONBERG, G
;
PATCHETT, AA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
PATCHETT, AA
;
LIESCH, JM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
LIESCH, JM
;
HENSENS, OD
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
HENSENS, OD
;
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MICROBIOL,RAHWAY,NJ 07065
SPRINGER, JP
.
SCIENCE,
1985,
230
(4722)
:177
-179
[8]
CYCLIC CHOLECYSTOKININ ANALOGS WITH HIGH SELECTIVITY FOR CENTRAL RECEPTORS
[J].
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